Claims Analysis
Total Claims: 11
Claim 1
Independent Claim
239 words
A compound selected from the group consisting of: a 1,2-benzisoxazole compound of the formula I: ##STR80## in which m is selected from the group consisting of: zero and the integers 1 to 5, n is 2, p is selected from the group consisting of: 0, 1 and 2, X, Y and Z, which may be identical or different, are each selected from the group consisting of a hydrogen atom, halogen atoms, linear and branched alkyl radicals having 1 to 6 carbon atoms, a trifluoromethyl radical, alkoxy radicals having 1 to 6 carbon atoms, alkylthio radicals having 1 to 6 carbon atoms and a hydroxyl radical, and a benzocyclobutenyl radical of formula A and an indanyl radical of formula B: ##STR81## in which R 1 and R 2 , which may be identical or different, are each selected from the group consisting of a hydrogen atom, halogen atoms, a trifluoromethyl radical, linear and branched alkyl radicals having 1 to 6 carbon atoms, alkoxy radicals having 1 to 6 carbon atoms, a hydroxyl radical, hydroxyalkyl radicals having 1 to 6 carbon atoms, and alkylthio radicals having 1 to 6 carbon atoms, and which together may form a methylenedioxy radical or an ethylenedioxy radical, and R 3 is selected from the group consisting of a hydrogen atom, linear and branched alkyl radicals having 1 to 6 carbon atoms, their optical isomers and their addition salts with a pharmaceutically-acceptable organic or inorganic acid.
Claim 2
Dependent Claim
239 words
A compound selected from the group consisting of: a 1,2-benzisoxazole compound of the formula I: ##STR80## in which m is selected from the group consisting of: zero and the integers 1 to 5, n is 2, p is selected from the group consisting of: 0, 1 and 2, X, Y and Z, which may be identical or different, are each selected from the group consisting of a hydrogen atom, halogen atoms, linear and branched alkyl radicals having 1 to 6 carbon atoms, a trifluoromethyl radical, alkoxy radicals having 1 to 6 carbon atoms, alkylthio radicals having 1 to 6 carbon atoms and a hydroxyl radical, and a benzocyclobutenyl radical of formula A and an indanyl radical of formula B: ##STR81## in which R 1 and R 2 , which may be identical or different, are each selected from the group consisting of a hydrogen atom, halogen atoms, a trifluoromethyl radical, linear and branched alkyl radicals having 1 to 6 carbon atoms, alkoxy radicals having 1 to 6 carbon atoms, a hydroxyl radical, hydroxyalkyl radicals having 1 to 6 carbon atoms, and alkylthio radicals having 1 to 6 carbon atoms, and which together may form a methylenedioxy radical or an ethylenedioxy radical, and R 3 is selected from the group consisting of a hydrogen atom, linear and branched alkyl radicals having 1 to 6 carbon atoms, their optical isomers and their addition salts with a pharmaceutically-acceptable organic or inorganic acid.
Claim 3
Dependent Claim
17 words
(RS)-3-[1-(Benzocyclobuten-1-ylmethyl)-4-piperidyl]-6-fluoro-1,2-benzisoxazole, as claimed in claim 1, and its addition salts with a pharmaceutically-acceptable inorganic or organic acid.
Claim 4
Dependent Claim
17 words
(+)-3-[1-(Benzocyclobuten-1-ylmethyl)-4-piperidyl]-6-fluoro-1,2-benzisoxazole, as claimed in claim 1, and its addition salts with a pharmaceutically-acceptable inorganic or organic acid.
Claim 5
Dependent Claim
17 words
(-)-3-[1-(Benzocyclobuten-1-ylmethyl)-4-piperidyl]-6-fluoro-1,2-benzisoxazole, as claimed in claim 1, and its addition salts with a pharmaceutically-acceptable inorganic or organic acid.
Claim 6
Dependent Claim
20 words
(RS)-3-[1-(2-Benzocyclobuten-1-ylethyl)-4-piperidyl]-6-fluoro-1,2-benzisoxazole, as claimed in claim 1, its optical isomers and its addition salts with a pharmaceutically-acceptable inorganic or organic acid.
Claim 7
Dependent Claim
20 words
(RS)-6-Fluoro-3-{1-[(1-methylbenzocyclobuten-1-yl)methyl]-4-piperidyl}-1,2-benzisoxazole, as claimed in claim 1, its optical isomers and its addition salts with a pharmaceutically-acceptable inorganic or organic acid.
Claim 8
Dependent Claim
20 words
(RS)-3-[1-(4,5-Dimethoxybenzocyclobuten-1-ylmethyl)-4-piperidyl]-6-fluoro-1,2-benzisoxazole, as claimed in claim 1, its optical isomers and its addition salts with a pharmaceutically-acceptable inorganic or organic acid.
Claim 9
Dependent Claim
20 words
(RS)-6-Fluoro-3-[1-(1-indanylmethyl)-4-piperidyl]-1,2-benzisoxazole, as claimed in claim 1, its optical isomers and its addition salts with a pharmaceutically-acceptable inorganic or organic acid.
Claim 10
Dependent Claim
33 words
A pharmaceutical composition useful in dopamine and serctonin antagonist containing as active principle an effective amount of a compound of claim 1, in combination or mixed with a pharmaceutically acceptable, vehicle or excipient.
Claim 11
Dependent Claim
46 words
A method for treating a living animal body afflicted with a disease requiring a dopamine and serctonin antagonist, comprising the step of administering to the said living animal an amount of a compound of claim 1 which is effective for the alleviation of the said condition.