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US4284788A Expired / Lapsed US ⏱️ 0.0 years remaining

Imidazolidone intermediates of biotin

Assignee: Hoffmann La Roche Inc
•
Filing: 1980-03-31
•
Granted: 1981-08-18
•
Expires: 2000-03-31
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Abstract

Abstract A process is disclosed for producing imidazolidone intermediates from 2H-chromene. The intermediates are useful for synthesizing biotin.

Inventors

  • 👤 Kraft Hohenlohe-Oehringen
  • 👤 Anton Fliri

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-09 20:13
CPC Classifications
C; C07; C07D; C07D491/00; C07D491/02; C07D491/04; C07D233/00; C07D233/04; C07D233/28; C07D233/30; C07D233/32; C07D495/00; C07D495/02; C07D495/04

Claims Analysis

Total Claims: 14
Claim 1
Independent Claim 11 words
A compound of the formula: ##STR16## wherein R 4a is azidosulphonyl.
Claim 2
Dependent Claim 11 words
A compound of the formula: ##STR16## wherein R 4a is azidosulphonyl.
Claim 3
Dependent Claim 29 words
A compound of the formula: ##STR17## wherein R 1 is hydrogen or a nitrogen protecting group selected from the group consisting of benzyl, alpha-lower alkyl substituted benzyl and allyl.
Claim 4
Dependent Claim 29 words
A compound of the formula: ##STR17## wherein R 1 is hydrogen or a nitrogen protecting group selected from the group consisting of benzyl, alpha-lower alkyl substituted benzyl and allyl.
Claim 5
Dependent Claim 10 words
The compound of claim 2 wherein R 1 is hydrogen.
Claim 6
Dependent Claim 26 words
The compound of claim 2 wherein R 1 is a nitrogen protecting group selected from the group consisting of benzyl, alpha-lower alkyl substituted benzyl and allyl.
Claim 7
Dependent Claim 12 words
The compound of claim 4 wherein the nitrogen protecting group is benzyl.
Claim 8
Dependent Claim 12 words
The compound of claim 4 wherein the nitrogen protecting group is allyl.
Claim 9
Dependent Claim 28 words
A compound of the formula: ##STR18## wherein R 1 is hydrogen or a nitrogen protecting group selected from the group consisting of benzyl, alpha-lower alkyl benzyl and allyl.
Claim 10
Dependent Claim 28 words
A compound of the formula: ##STR18## wherein R 1 is hydrogen or a nitrogen protecting group selected from the group consisting of benzyl, alpha-lower alkyl benzyl and allyl.
Claim 11
Dependent Claim 10 words
The compound of claim 7 wherein R 1 is hydrogen.
Claim 12
Dependent Claim 26 words
The compound of claim 7 wherein R 1 is a nitrogen protecting group selected from the group consisting of benzyl, alpha-lower alkyl substituted benzyl and allyl.
Claim 13
Dependent Claim 12 words
The compound of claim 9 wherein the nitrogen protecting group is benzyl.
Claim 14
Dependent Claim 12 words
The compound of claim 9 wherein the nitrogen protecting group is allyl.

References Cited (Backward Citations)

DE2508831A1 Cited
US4044020A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1984-08-17 1985-02-16 1985-08-18 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1988-08-17 1989-02-16 1989-08-18 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1992-08-17 1993-02-16 1993-08-18 $7700.00 Window Closed / Lapsed

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