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N-(1-Substituted-3-pyrrolidinyl)benzamides

Assignee: Wyeth LLC
•
Filing: 1976-12-06
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Granted: 1981-07-21
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Expires: 1996-12-06
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Abstract

Abstract N-(1-Substituted-3-pyrrolidinyl)benzamides of the formula ##STR1## wherein R is cycloalkyl or phenyllower-alkyl; R 1 is hydrogen or lower alkyl of 1 to 8 carbon atoms; R 2 is acetamido, amino, methylamino, dimethylamino, benzyloxy, halogen, lower alkoxy, methylmercapto, nitro, cyano, hydroxy, sulfamoyl, bis(methylsulfonyl)amino, methylsulfonylamino, aminomethyl or acetylaminomethyl and can be the same or different; n is an integer from one to three inclusive with the proviso that when R 2 is amino, nitro, halogen or lower alkoxy, n is greater than one, and pharmaceutically acceptable acid addition salts thereof are disclosed.

Inventors

  • 👤 Albert D. Cale, Jr.
  • 👤 Charles A. Leonard

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-07 22:41
CPC Classifications
C; C07; C07D; C07D207/00; C07D207/02; C07D207/04; C07D207/10; C07D207/14

Claims Analysis

Total Claims: 8
Claim 1
Independent Claim 1 words
N-(1-cyclohexyl-3-pyrrolidinyl)-4-acetamidobenzamide.
Claim 2
Dependent Claim 1 words
N-(1-cyclohexyl-3-pyrrolidinyl)-4-acetamidobenzamide.
Claim 3
Dependent Claim 1 words
N-(1-cyclohexyl-3-pyrrolidinyl)-2-methoxy-5-sulfamoylbenzamide.
Claim 4
Dependent Claim 1 words
N-(1-cyclohexyl-3-pyrrolidinyl)-2-methoxy-5-sulfamoylbenzamide.
Claim 5
Dependent Claim 5 words
The fumarate salt of N-(1-cyclohexyl-3-pyrrolidinyl)-2-methoxy-4-amino-5-chlorobenzamide.
Claim 6
Dependent Claim 5 words
The fumarate salt of N-(1-cyclohexyl-3-pyrrolidinyl)-2-methoxy-4-amino-5-chlorobenzamide.
Claim 7
Dependent Claim 1 words
N-(1-cyclohexyl-3-pyrrolidinyl)-2-methoxy-4-amino-5-chlorobenzamide.
Claim 8
Dependent Claim 1 words
N-(1-cyclohexyl-3-pyrrolidinyl)-2-methoxy-4-amino-5-chlorobenzamide.

References Cited (Backward Citations)

US3342826A Cited
US3577440A Cited
US4013670A Cited
US4002757A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1984-07-20 1985-01-19 1985-07-21 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1988-07-20 1989-01-19 1989-07-21 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1992-07-20 1993-01-19 1993-07-21 $7700.00 Window Closed / Lapsed

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