Triazolylbenzophenone derivatives and production thereof
Abstract
Abstract Triazolylbenzophenone derivatives of the formula: ##STR1## (wherein R represents hydrogen, C 1 -C 6 alkyl, C 1 -C 6 halo-alkyl, the group --(CH 2 ) n --X--R 5 , or the group ##STR2## R 5 represents hydrogen, C 1 -C 6 alkyl, C 2 -C 6 alkenyl, C 2 -C 6 alkynyl, C 6 -C 10 aryl, or C 2 -C 8 acyl; X represents sulfur or oxygen; n represents 0, 1, 2, or 3; R 6 and R 7 each represents hydrogen or C 1 -C 6 alkyl; or the group ##STR3## represents pyrrolidino, piperidino, morpholino, or γ-methylpiperazino; R 1 represents hydrogen or halogen; R 2 represents halogen, nitro, or trifluoromethyl; R 3 represents C 1 -C 6 alkyl, C 1 -C 6 halo-alkyl, C 1 -C 6 azido-alkyl, C 6 -C 10 aryl, C 2 -C 8 acyl, or the group ##STR4## R 4 and R 8 each represents hydrogen, C 1 -C 6 alkyl, or C 7 -C 10 aralkyl; R 9 represents hydrogen or C 1 -C 6 alkyl; R 10 represents hydrogen, C 1 -C 6 alkyl, C 7 -C 10 aralkyl, or C 2 -C 11 α-amino-acyl; or the group ##STR5## represents phthalimido, pyrrolidino, piperidino, morpholino, or γ-methylpiperazino) and their pharmaceutically acceptable acid addition salts, useful as anxiolytics, sedatives, hypnotics, anticonvulsants, muscle relaxants, antidepressants, their synthetic intermediates, and their preparation.
Inventors
- 👤 Kentaro Hirai
- 👤 Toshio Fujishita
- 👤 Teruyuki Ishiba
- 👤 Hirohiko Sugimoto
Bibliographic Details
Claims Analysis
Total Claims: 2References Cited (Backward Citations)
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