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US4065473A
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Intermediates in the preparation of 2,3,4,5-tetrahydro-1H-3-benzazepines
Assignee: Hoffmann La Roche Inc
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Filing: 1975-06-20
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Granted: 1977-12-27
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Expires: 1995-06-20
Abstract
Abstract A process for the preparation of heterocyclic compounds containing one nitrogen atom and novel 2,3,4,5-tetrahydro-1H-3-benzazepines prepared by this process are disclosed. The resulting heterocyclic compounds, including the novel 2,3,4,5-tetrahydro-1H-3-benzazepine derivatives, exhibit analgesic, appetite suppressant, and anti-edema activity.
Inventors
- 👤 Arnold Brossi
- 👤 Benjamin Pecherer
- 👤 Robert Sunbury
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-04 10:11
CPC Classifications
C; C07; C07D; C07D209/00; C07D209/02; C07D209/44; C07D209/48; C07D491/00; C07D491/02; C07D491/04; C07D491/056
Claims Analysis
Total Claims: 4
Claim 1
Independent Claim
58 words
A compound selected from the group consisting of compounds of the formula ##STR18## wherein R 2 and R 3 taken together signify methylenedioxy; R 4 signifies hydrogen, lower alkyl, carboxy, aryl or aryl substituted by a member selected from the group consisting of halogen, lower alkyl, nitro, or trifluoromethyl; n is 1 or 2; and X is acetyl.
Claim 2
Dependent Claim
58 words
A compound selected from the group consisting of compounds of the formula ##STR18## wherein R 2 and R 3 taken together signify methylenedioxy; R 4 signifies hydrogen, lower alkyl, carboxy, aryl or aryl substituted by a member selected from the group consisting of halogen, lower alkyl, nitro, or trifluoromethyl; n is 1 or 2; and X is acetyl.
Claim 3
Dependent Claim
2 words
N-6-Chloromethyl-3,4-methylenedioxyphenethyl) acetamide.
Claim 4
Dependent Claim
2 words
N-6-Chloromethyl-3,4-methylenedioxyphenethyl) acetamide.
References Cited (Backward Citations)
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Cited
US3146266A
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US3801601A
Cited
US3498988A
Cited
US3520904A
Cited
US3689557A
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US3784640A
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USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1980-12-26 | 1981-06-27 | 1981-12-27 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1984-12-26 | 1985-06-27 | 1985-12-27 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1988-12-26 | 1989-06-27 | 1989-12-27 | $7700.00 | Window Closed / Lapsed |