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α-Aminomethylbenzyl alcohol derivatives

Assignee: Astellas Pharma Inc
•
Filing: 1974-05-07
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Granted: 1976-11-30
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Expires: 1994-05-07
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Abstract

Abstract Novel alpha -aminomethylbenzyl alcohol derivatives, particularly alpha -aminoethyl-3-substituted amino-4-hydroxybenzyl alcohol derivatives. The compounds of this invention are useful as bronchodilating agents.

Inventors

  • 👤 Masuo Murakami
  • 👤 Kozo Takahashi
  • 👤 Toshiyasu Mase
  • 👤 Kiyoshi Murase
  • 👤 Hisashi Ida

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-06 08:27
CPC Classifications
A; A61; A61K; A61K31/00; A61K31/16; A61K31/165; A61K31/13; A61K31/135; A61K31/185; A61K31/205; C; C07; C07C; C07C215/00; C07C215/74; C07C215/76; C07C233/00; C07C233/01; C07C233/16; C07C237/00

Claims Analysis

Total Claims: 5
Claim 1
Independent Claim 23 words
A compound selected from the group consisting of 3-formylamino-4-hydroxy-α-[N-(1-methyl-2-p-methoxyphenylethyl)aminomethyl]benzyl alcohol of the formula: ##SPC24## and the pharmacologically acceptable non-toxic acid addition salts thereof.
Claim 2
Dependent Claim 23 words
A compound selected from the group consisting of 3-formylamino-4-hydroxy-α-[N-(1-methyl-2-p-methoxyphenylethyl)aminomethyl]benzyl alcohol of the formula: ##SPC24## and the pharmacologically acceptable non-toxic acid addition salts thereof.
Claim 3
Dependent Claim 12 words
A compound according to claim 1 which is 3-formylamino-4-hydroxy-α-[N-(1-methyl-2-p-methoxyphenylethyl)aminomethyl]benzyl alcohol 1/2 fumarate.
Claim 4
Dependent Claim 19 words
A compound according to claim 1 which is 3-formylamino-4-hydroxy-α-[N-(1-methyl-2-p-methoxyphenylethyl)aminomethyl]benzyl alcohol 1/2 fumarate showing melting point (decomposition) of 138°-140° C.
Claim 5
Dependent Claim 20 words
A compound according to claim 1 which is 3-formylamino-4-hydroxy-α-[N-(1-methyl-2-p-methoxyphenylethyl)aminomethyl]-benzyl alcohol of 1/2 fumarate showing melting point (decomposition) of 154°-155° C.

References Cited (Backward Citations)

US2393820A Cited
US3644520A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1979-11-30 1980-05-31 1980-11-30 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1983-11-30 1984-05-31 1984-11-30 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1987-11-30 1988-05-31 1988-11-30 $7700.00 Window Closed / Lapsed

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