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US3966730A
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Pyrimidin(4)-yl-(thiono)-(thiol)-phosphoric-(phosphonic)-acid esters
Assignee: Bayer AG
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Filing: 1974-08-22
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Granted: 1976-06-29
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Expires: 1994-08-22
Abstract
Abstract Pyrimidin(4)-yl-(thiono)-phosphoric-(phosphonic) acid esters and ester amides of the formula IN WHICH R1 is hydrogen, alkyl, cycloalkyl, alkenyl, alkynyl, aryl or aralkyl, R2 is hydrogen, alkyl, alkoxy, alkylmercapto, alkylcarbonyl, alkoxycarbonyl, halogen, nitrile or thiocyanato, R3 is hydrogen, alkyl, aryl or alkoxycarbonylalkyl, or R2 is R3 conjointly form an alkylene bridge which forms a 5-membered to 7-membered ring with the adjoining carbon atoms, R4 is alkyl or alkoxyalkyl, R5 is alkyl, alkoxy, alkylmercapto, alkylamino, or aryl, and X is oxygen or sulfur, WHICH POSSESS INSECTICIDAL, ACARICIDAL AND NEMATOCIDAL PROPERTIES.
Inventors
- 👤 Wolfgang Hofer
- 👤 Fritz Maurer
- 👤 Hans-Jochem Riebel
- 👤 Lother Rohe
- 👤 Wolfgang Behrenz
- 👤 Ingeborg Hammann
- 👤 Wilhelm Stendel
- 👤 Bernhard Homeyer
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-10-30 15:10
CPC Classifications
C; C07; C07F; C07F9/00; C07F9/02; C07F9/547; C07F9/645; C07F9/6509; C07F9/6512
Claims Analysis
Total Claims: 4
Claim 1
Independent Claim
233 words
A pyrimidin(4)-yl-(thiono)-(thiol)-phosphoric-(phosphonic) acid ester or ester-amide of the formula ##SPC11## in which R 1 is straight-chain or branched alkyl with 1 to 20 carbon atoms, cycloalkyl with 5 to 7 carbon atoms, alkenyl or alkynyl with 2 to 6 carbon atoms or aralkyl with 6 to 10 carbon atoms in the aryl moiety and 1 to 2 carbon atoms in the alkyl moiety, R 2 is hydrogen, straight-chain or branched alkyl with 1 to 4 carbon atoms, alkoxy with 1 to 4 carbon atoms, alkylmercapto with 1 to 4 carbon atoms, alkylcarbonyl or alkoxycarbonyl with 1 to 4 carbon atoms in the alkyl or alkoxy moiety, halogen or nitrile, R 3 is hydrogen, straight-chain or branched alkyl with 1 to 6 carbon atoms, or alkoxycarbonylalkyl with 1 to 4 carbon atoms in the alkoxy radical and 1 to 2 carbon atoms in the alkyl radical, or R 2 and R 3 conjointly form an alkylene bridge which forms a 5-membered to 7-membered ring with the adjoining carbon atoms, R 4 is straight-chain or branched alkyl with 1 to 12 carbon atoms or alkoxyalkyl with 1 to 12 carbon atoms in the alkyl radical and 1 to 4 carbon atoms in the alkoxy radical, R 5 is straight-chain or branched alkyl, alkoxy or alkylmercapto with 1 to 6 carbon atoms or aryl with 6 to 10 carbon atoms, and X is oxygen or sulfur
Claim 2
Dependent Claim
233 words
A pyrimidin(4)-yl-(thiono)-(thiol)-phosphoric-(phosphonic) acid ester or ester-amide of the formula ##SPC11## in which R 1 is straight-chain or branched alkyl with 1 to 20 carbon atoms, cycloalkyl with 5 to 7 carbon atoms, alkenyl or alkynyl with 2 to 6 carbon atoms or aralkyl with 6 to 10 carbon atoms in the aryl moiety and 1 to 2 carbon atoms in the alkyl moiety, R 2 is hydrogen, straight-chain or branched alkyl with 1 to 4 carbon atoms, alkoxy with 1 to 4 carbon atoms, alkylmercapto with 1 to 4 carbon atoms, alkylcarbonyl or alkoxycarbonyl with 1 to 4 carbon atoms in the alkyl or alkoxy moiety, halogen or nitrile, R 3 is hydrogen, straight-chain or branched alkyl with 1 to 6 carbon atoms, or alkoxycarbonylalkyl with 1 to 4 carbon atoms in the alkoxy radical and 1 to 2 carbon atoms in the alkyl radical, or R 2 and R 3 conjointly form an alkylene bridge which forms a 5-membered to 7-membered ring with the adjoining carbon atoms, R 4 is straight-chain or branched alkyl with 1 to 12 carbon atoms or alkoxyalkyl with 1 to 12 carbon atoms in the alkyl radical and 1 to 4 carbon atoms in the alkoxy radical, R 5 is straight-chain or branched alkyl, alkoxy or alkylmercapto with 1 to 6 carbon atoms or aryl with 6 to 10 carbon atoms, and X is oxygen or sulfur
Claim 3
Dependent Claim
17 words
The compound according to claim 1 wherein such compound is O-methyl-O-[2-methoxy-6-methyl-pyrimidyl-(4)]-ethanethionophosphonic acid ester of the formula ##SPC12##
Claim 4
Dependent Claim
17 words
The compound according to claim 1 wherein such compound is O-methyl-O-[2-ethoxy-6-methyl-pyrimidyl-(4)]-ethanethionophosphonic acid ester of the formula ##SPC13##
References Cited (Backward Citations)
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1979-06-29 | 1979-12-29 | 1980-06-29 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1983-06-29 | 1983-12-29 | 1984-06-29 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1987-06-29 | 1987-12-29 | 1988-06-29 | $7700.00 | Window Closed / Lapsed |