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Carbostyril derivatives and process for preparing the same

Assignee: Otsuka Pharmaceutical Co Ltd
•
Filing: 1973-12-14
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Granted: 1976-04-27
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Expires: 1993-12-14
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Abstract

Abstract 2-Hydroxy-3-alkylaminopropoxycarbostyrils represented by the formula (I) ##SPC1## wherein R represents a straight or branched chain alkyl group having 1 to 4 carbon atoms useful as β-adrenergic blocking agents and a process for preparing the same are disclosed.

Inventors

  • 👤 Kazuyuki Nakagawa
  • 👤 Shiro Yoshizaki
  • 👤 Nanami Murakami
  • 👤 Hideo Mori

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-05 23:11
CPC Classifications
C; C07; C07D; C07D215/00; C07D215/02; C07D215/16; C07D215/20; C07D215/22; C07D215/227; A; A61; A61P; A61P9/00; A61P9/06; A61P9/08; A61P9/10; C07D215/24; C07D215/26

Claims Analysis

Total Claims: 7
Claim 1
Independent Claim 35 words
A 5- or 8- (2-Hydroxy-3-alkylamino)propoxycarbostyril compound represented by the formula (I): ##SPC4## wherein R represents a straight or branched alkyl group having 1 to 4 carbon atoms, and the pharmaceutically acceptable acid addition salts thereof.
Claim 2
Dependent Claim 35 words
A 5- or 8- (2-Hydroxy-3-alkylamino)propoxycarbostyril compound represented by the formula (I): ##SPC4## wherein R represents a straight or branched alkyl group having 1 to 4 carbon atoms, and the pharmaceutically acceptable acid addition salts thereof.
Claim 3
Dependent Claim 5 words
5-(2-Hydroxy-3-isopropylamino)propoxycarbostyril according to claim 1.
Claim 4
Dependent Claim 5 words
5-(2-Hydroxy-3-tert-butylamino)propoxycarbostyril according to claim 1.
Claim 5
Dependent Claim 5 words
8-(2-Hydroxy-3-tert-butylamino)propoxycarbostyril according to claim 1.
Claim 6
Dependent Claim 5 words
8-(2-Hydroxy-3-isopropylamino)propoxycarbostyril according to claim 1.
Claim 7
Dependent Claim 5 words
8-(2-Hydroxy-3-sec-butylamino)propoxycarbostyril according to claim 1.

References Cited (Backward Citations)

GB1058822A Cited
US3340266A Cited
GB1047927A Cited
GB1079989A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1979-04-27 1979-10-27 1980-04-27 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1983-04-27 1983-10-27 1984-04-27 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1987-04-27 1987-10-27 1988-04-27 $7700.00 Window Closed / Lapsed

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