US3933811A
Expired / Lapsed
US
⏱️ 0.0 years remaining
N-aminomethyl-2-amino(and 2-amino-methyl)-2-(2-quinolyl)-thioacetamides
Assignee: GlaxoSmithKline LLC
•
Filing: 1974-09-18
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Granted: 1976-01-20
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Expires: 1994-09-18
Abstract
Abstract The compounds are N-aminomethyl-2-amino(and 2-aminomethyl)-2-heterocyclic-thioacetamides which are inhibitors of gastric acid secretion.
Inventors
- 👤 L. Martin Brenner
- 👤 Bernard Loev
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-08 19:04
CPC Classifications
C; C07; C07D; C07D295/00; C07D295/04; C07D295/12; A; A61; A61K; A61K31/00; A61K31/33; A61K31/395; A61K31/435; A61K31/44; C07D239/00; C07D239/02; C07D239/24; C07D239/26; C07D241/00; C07D241/02; C07D241/10; C07D241/12; C07D413/00; C07D413/02; C07D413/12
Claims Analysis
Total Claims: 5
Claim 1
Independent Claim
40 words
A compound of the formula: ##EQU5## in which m is 0 or 1; R 1 is 2-quinolyl; and R 2 and R 3 are di-lower alkylamino, N-lower Alkyl-N-phenylamino, piperidino, pyrrolidino or morpoholino or a pharmaceutically acceptable acid addition salt thereof.
Claim 2
Dependent Claim
40 words
A compound of the formula: ##EQU5## in which m is 0 or 1; R 1 is 2-quinolyl; and R 2 and R 3 are di-lower alkylamino, N-lower Alkyl-N-phenylamino, piperidino, pyrrolidino or morpoholino or a pharmaceutically acceptable acid addition salt thereof.
Claim 3
Dependent Claim
40 words
A compounds of claim 1 in which m is 0 or 1 and R 2 is dimethylamino, diethylamino, piperidino or pyrrolidino or m is 1 and R 2 is morpholino, and R 3 is di-lower alkylamino, piperidino, pyrrolidino or morpholino.
Claim 4
Dependent Claim
9 words
A compound of claim 1, said compound being 3-morpholino-N-morpholinomethyl-2-(2-quinolyl)thiopropanamide.
Claim 5
Dependent Claim
9 words
A compound of claim 1, said compound being 2-dimethylamino-N-morpholinomethyl-2-(2-quinolyl)thioacetamide.
References Cited (Backward Citations)
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Cited
US3876645A
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US3660592A
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US3749728A
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US3880860A
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US3740409A
Cited
US3882126A
Cited
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Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1979-01-19 | 1979-07-21 | 1980-01-20 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1983-01-19 | 1983-07-21 | 1984-01-20 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1987-01-19 | 1987-07-21 | 1988-01-20 | $7700.00 | Window Closed / Lapsed |