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US3875154A Expired / Lapsed US ⏱️ 0.0 years remaining

Certain 5-thia-1-azabicyclo{8 4.2.0{9 octenes

Assignee: University of California
•
Filing: 1973-12-17
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Granted: 1975-04-01
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Expires: 1993-12-17
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Abstract

Abstract A process for preparing lactams, particularly 1azabicyclo(4.2.0)octanes, 1-azabicyclo(3.2.0)heptanes, 4-thia-1azabicyclo(3.2.0)heptanes and 5-thia-1-azabicyclo (4.2.0)octenes, which comprises subjecting a cyclic Alpha -ketoamide to an oxidizing agent to form a carboxyl substituted lactam structure. The oxidant is preferably periodate, in an aqueous solution, at pH 5-9 and room temperature. The novel products obtained from the process are useful intermediates in the preparation of antimicrobial agents. The cyclic Alpha -ketoamide starting materials are also novel.

Inventors

  • 👤 Henry Rapoport

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-03 20:29
CPC Classifications
C; C07; C07D; C07D499/00

Claims Analysis

Total Claims: 3
Claim 1
Independent Claim 5 words
A COMPOUND OF THE FORMULA:
Claim 2
Dependent Claim 5 words
A COMPOUND OF THE FORMULA:
Claim 3
Dependent Claim 11 words
A compound according to claim 1 in which R is hydrogen.

References Cited (Backward Citations)

US3534029A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1978-03-31 1978-09-30 1979-04-01 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1982-03-31 1982-09-30 1983-04-01 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1986-03-31 1986-09-30 1987-04-01 $7700.00 Window Closed / Lapsed

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