Patent US4020393A successfully refreshed from Google Patents.
Patent US3870709A successfully refreshed from Google Patents.
← Back to Patent Explorer
US3870709A Expired / Lapsed US ⏱️ 0.0 years remaining

6-(alpha-(ome ga-guanidinoalkanoylamido)acylamido)penicillanic acids

Assignee: Pfizer Inc
•
Filing: 1972-02-22
•
Granted: 1975-03-11
•
Expires: 1992-02-22
📄 Original PDF 🌐 Google Patents 🔄 Sync Now

Abstract

Abstract 6-( Alpha -( omega GUANIDINOALKANOYLAMIDO)ACYLAMIDO)PENICILLANIC ACIDS, THE NONTOXIC SALTS AND ESTERS THEREOF ARE USEFUL AS ANTIBACTERIAL AGENTS, THERAPEUTIC AGENTS IN ANIMALS, INCLUDING MAN, OF PARTICULAR VALUE AGAINST GRAM-NEGATIVE BACTERIA, AND AS ANIMAL FEED NUTRITIONAL SUPPLEMENTS.

Inventors

  • 👤 Ernest S Hamanaka

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-10-26 20:08
CPC Classifications
C; C07; C07D; C07D499/00; C07D499/21; C07D499/44; C07D499/48; C07D499/58; C07D499/64

Claims Analysis

Total Claims: 15
Claim 1
Independent Claim 5 words
A compound of the formula
Claim 2
Dependent Claim 5 words
A compound of the formula
Claim 3
Dependent Claim 5 words
A COMPOUND OF THE FORMULA
Claim 4
Dependent Claim 5 words
A COMPOUND OF THE FORMULA
Claim 5
Dependent Claim 25 words
A compound according to claim 1 wherein R1 is phenyl; each of R2, R3, R4, R5, R6 and R is hydrogen; and X is alkylene.
Claim 6
Dependent Claim 30 words
A compound according to claim 1 wherein R1 is phenyl; each of R2, R3, R4, R5 and R6 is hydrogen; R is lower alkanoyloxy lower alkyl; and X is alkylene.
Claim 7
Dependent Claim 25 words
A compound according to claim 1 wherein R1 is phenyl; each of R2, R3, R4, R5, R6 and R is hydrogen; and X is phenylene.
Claim 8
Dependent Claim 25 words
A compound according to claim 1 wherein R1 is phenyl; each of R2, R3, R4, R5, R6 and R is hydrogen; and X is phenylenemethylene.
Claim 9
Dependent Claim 27 words
A compound according to claim 1 wherein R1 is phenyl; R3 is methyl; each of R2, R4, R5, R6 and R is hydrogen; and X is alkylene.
Claim 10
Dependent Claim 40 words
A compound according to claim 1 wherein R1 is phenyl, R3 and R5 when taken together with the guanidino moiety to which they are attached are imidazolidino; X is methylene; and each of R2, R4, R6 and R is hydrogen.
Claim 11
Dependent Claim 27 words
A compound according to claim 1 wherein R1 is 1,4-cyclohexadienyl; each of R2, R3, R4, R6 and R is hydrogen; R5 is methyl; and X is methylene.
Claim 12
Dependent Claim 25 words
The compound according to claim 2 wherein R1 is phenyl, each of R2, R3, R4, R5, R6 and R is hydrogen; and X is methylene.
Claim 13
Dependent Claim 27 words
The compound according to claim 3 wherein R1 is phenyl, each of R2, R3, R4, R5 and R6 is hydrogen; R is pivaloyloxymethyl; and X is methylene.
Claim 14
Dependent Claim 25 words
The compound according to claim 4 wherein R1 is phenyl; each of R2, R3, R4, R5, R6 and R is hydrogen; and X is 1,4-phenylene.
Claim 15
Dependent Claim 25 words
The compound according to claim 5 wherein R1 is phenyl; each of R2, R3, R4, R5, R6 and R is hydrogen; and X is 1,4-phenylenemethylene.

References Cited (Backward Citations)

US3579501A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1978-03-10 1978-09-09 1979-03-11 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1982-03-10 1982-09-09 1983-03-11 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1986-03-10 1986-09-09 1987-03-11 $7700.00 Window Closed / Lapsed

Assigned Categories & Tags

No categories assigned to this patent yet.

Assign Category Tag