US3853835A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Alkyl esters of aspartyl aliphatic amino acid dipeptides
Assignee: Nutrasweet Co
•
Filing: 1972-10-30
•
Granted: 1974-12-10
•
Expires: 1992-10-30
Abstract
Abstract Coupling of the appropriate (S)-aspartic acid derivative with an aliphatic amino acid alkyl ester followed by hydrogenolysis of the protecting groups affords the corresponding (S)-aspartyl-(R)(aliphatic-) amino acid alkyl esters, which exhibit potent sweetening properties.
Inventors
- 👤 R Mazur
- 👤 J Schlatter
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-10-26 09:37
CPC Classifications
C; C07; C07K; C07K5/00; C07K5/04; C07K5/06; C07K5/06104; C07K5/06113; A; A23; A23L; A23L27/00; A23L27/30; A23L27/31; A23L27/32; Y; Y02; Y02P; Y02P20/00; Y02P20/50; Y02P20/55; Y10; Y10S; Y10S530/00; Y10S530/801
Claims Analysis
Total Claims: 13
Claim 1
Independent Claim
5 words
A COMPOUND OF THE FORMULA
Claim 2
Dependent Claim
5 words
A COMPOUND OF THE FORMULA
Claim 3
Dependent Claim
50 words
As in claim 1, a compound of the formula v,90/8 wherein R, R'' and R'''' are lower alkyl radicals containing less than four carbon atoms with the provision that, when R'' and R'''' are dissimilar, the carbon atom to which R'' and R'''' are attached possesses the (R) stereochemical configuration.
Claim 4
Dependent Claim
9 words
As in claim 1, a compound of the formula
Claim 5
Dependent Claim
11 words
As in claim 1, the compound which is (S)-aspartyl-(R)-alanine n-propyl ester.
Claim 6
Dependent Claim
11 words
As in claim 1, the compound which is (S)-aspartyl-(R)-alanine isopropyl ester.
Claim 7
Dependent Claim
11 words
As in claim 1, the compound which is (S)-aspartyl-(R)-alanine methyl ester.
Claim 8
Dependent Claim
14 words
As in claim 1, the compound which is (S)-aspartyl-(R)- Alpha -aminobutyric acid isopropyl ester.
Claim 9
Dependent Claim
11 words
As in claim 1, the compound which is (S)-aspartyl-(R)-valine isopropyl ester.
Claim 10
Dependent Claim
13 words
As in claim 1, the compound which is (S)-aspartyl- Alpha -methylalanine isopropyl ester.
Claim 11
Dependent Claim
13 words
As in claim 1, the compound which is (S)-aspartyl- Alpha -methylalanine ethyl ester.
Claim 12
Dependent Claim
11 words
As in claim 1, the compound which is (S)-aspartyl-(R)-isovaline isopropyl ester.
Claim 13
Dependent Claim
13 words
As in claim 1, the compound which is (S)-aspartyl-(R)- Alpha -methylvaline isopropyl ester.
References Cited (Backward Citations)
US3714139A
Cited
US3695898A
Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1977-12-09 | 1978-06-10 | 1978-12-10 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1981-12-09 | 1982-06-10 | 1982-12-10 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1985-12-09 | 1986-06-10 | 1986-12-10 | $7700.00 | Window Closed / Lapsed |