Ureidophenylisothioureas

Abstract

Abstract UREIDOPHENYLISOTHIOUREAS OF THE FORMULA 1-(R-OOC-NH-C(-S-R"")=N-),2-(R"-N(-R''")-CO-N(-R'')-),(X)N- BENZENE IN WHICH N IS 0, 1 OR 2 X IS HALOGEN, LOWER ALKYL OR ALKOXY, R IS LOWER ALKYL, R'' AND R" ARE EACH HYDROGEN OR LOWER ALKYL, R"'' IS HYDROGEN; ALKYL WITH 1 TO 18 CARBON ATOMS OPTIONALLY SUBSTITUTED BY HALOGEN, NITRILE, LOWER ALKOXY OR LOWER ALKOXYCARBONYL; CYCLOALKYL WITH 5 TO 8 CARBON ATOMS; ARALKYL OPTIONALLY SUBSTITUTED IN THE ARYL MOIETY BY HALOGEN, LOWER ALKYL OR ALKOXY; PHENYL OPTIONALLY SUBSTITUTED BY HALOGEN, LOWER ALKYL OR ALKOXY; ACYL WITH UP TO 18 CARBON ATOMS OPTIONALLY SUBSTITUTED BY HALOGEN OR LOWER ALKOXY; AROYL OPTIONALLY SUBSTITUTED BY HALOGEN, LOWER ALKYL OR ALKOXY; ALKYSULFONYL; ARYLSULFONYL OPTIONALLY SUBSTITUTED BY HALOGEN, AMINO, LOWER ALKYL OR ALKOXY; OR DI-LOWER ALKYLAMINO; OR R" AND R"'', TOGETHER WITH THE BONDING NITROGEN ATOM, FORM A HETEROCYCLIC RING WITH 4 TO 7 CARBON ATOMS, WHICH RING OPTIONALLY CONTAINS OXYGEN OR SULFUR AS FURTHER HETERO-ATOMS, AND R"" IS ALKYL WITH 1 TO 12 CARBON ATOMS, CYCLOALKYL WITH 3 TO 8 CARBON ATOMS, ALKENYL WITH UP TO 12 CARBON ATOMS OR ARALKYL OPTIONALLY SUBSTITUTED IN THE ARYL MOIETY BY HALOGEN, LOWER ALKYL OR ALKOXY, WHICH POSSESS FUNGICIDAL, INSECTICIDAL ACARICIDAL, ANTIBACTERIAL AND GROWTH-REGULATING PROPERTIES.

Inventors

• 👤 A Widdig
• 👤 F Grewe
• 👤 H Kaspers
• 👤 E Kuhle
• 👤 H Scheinpflug
• 👤 P Frohberger

Bibliographic Details