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1-substituted-5-nitroimidazol-2-ylalkyl-(n-substituted)-carbamates

Assignee: Merck and Co Inc
•
Filing: 1971-11-12
•
Granted: 1973-09-25
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Expires: 1991-11-12
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Abstract

Abstract 1-Substituted-5-nitroimidazol-2-ylalkyl carbamates containing Nacyl substituents, and acid addition salts thereof are prepared from 1-substituted-5-nitroimidazoles having at the 2-position of the imidazole ring an hydroxyalkyl, mercaptoalkyl, haloalkyl, halo-carbonylalkyl or halothiocarbonyloxyalkyl radical. The 1substituted-5-nitroimidazol-2-ylalkyl-(N-substituted)-carbamates are useful in the treatment of parasitic diseases. Antiparasitic compositions in which the active ingredient is a 1-substitutedimidazol-2-ylalkyl-(N-substituted)-carbamate are also provided.

Inventors

  • 👤 J Carlson
  • 👤 D Hoff
  • 👤 C Rooney

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-10-30 18:44
CPC Classifications
C; C07; C07D; C07D233/00; C07D233/54; C07D233/66; C07D233/91; C07D233/92; C07D233/94; A; A23; A23K; A23K20/00; A23K20/10; A23K20/116; A23K20/137

Claims Analysis

Total Claims: 8
Claim 1
Independent Claim 10 words
The compound of claim 1 in which R1 is methyl.
Claim 2
Dependent Claim 10 words
The compound of claim 2 in which Q is methylene.
Claim 3
Dependent Claim 13 words
The compound of claim 3 in which both A and M are oxygen.
Claim 4
Dependent Claim 10 words
The compound of claim 4 in which R4 is loweralkanoyl.
Claim 5
Dependent Claim 10 words
The compound of claim 5 in which R4 is acetyl.
Claim 6
Dependent Claim 10 words
The compound of claim 5 in which R4 is formyl.
Claim 7
Dependent Claim 10 words
The compound of claim 4 in which R4 is chloroacetyl.
Claim 8
Dependent Claim 10 words
The compound of claim 4 in which R4 is benzoyl.

References Cited (Backward Citations)

US3378552A Cited
US3325507A Cited
US3299090A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1976-09-24 1977-03-26 1977-09-25 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1980-09-24 1981-03-26 1981-09-25 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1984-09-24 1985-03-26 1985-09-25 $7700.00 Window Closed / Lapsed

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