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US3682930A
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US
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4(1-alkyl-4-piperidylidine)-4h-benzo {84,5{9 {0 cyclohepta {8 1,2{14 6{9
Assignee: Individual
•
Filing: 1971-03-03
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Granted: 1972-08-08
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Expires: 1991-03-03
Abstract
Abstract The present invention concerns novel compounds of the formula, WHEREIN R1 is hydrogen, halogen, or alkoxy of one to four carbon atoms, R2 is alkyl of one to four carbon atoms, and -A-B- is -CO-CH2-CO- or -CO-CH2-, and pharmaceutically acceptable acid addition salts thereof. The compounds are histaminolytics. Compounds wherein -A-B- is CO-CH2- are antaminics, i.e. aside from histaminolytic properties, they possess serotonin - antagonistic and anticholinergic properties.
Inventors
- 👤 Jean-Pierre Bourquin
- 👤 Gustav Schwarb
- 👤 Erwin Waldvogel
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-05 15:05
CPC Classifications
C; C07; C07D; C07D333/00; C07D333/02; C07D333/04; C07D333/06; C07D333/24; C07D333/50; C07D333/78; C07D333/80
Claims Analysis
Total Claims: 19
Claim 1
Independent Claim
9 words
The compound of claim 1, which is 4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen-9(10H) -one.
Claim 2
Dependent Claim
9 words
The compound of claim 1, which is 4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen-10(9H) -one.
Claim 3
Dependent Claim
9 words
The compound of claim 1, which is 4-(1-ethyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen-9(10H) -one.
Claim 4
Dependent Claim
9 words
The compound of claim 1, which is 4-(1-ethyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen-10(9H) -one.
Claim 5
Dependent Claim
9 words
The compound of claim 1, which is 4-(1-isopropyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen -10(9H)-one.
Claim 6
Dependent Claim
9 words
The compound of claim 1, which is 4-(1n-butyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen-10(9H) -one.
Claim 7
Dependent Claim
9 words
The compound of claim 1, which is 6-chloro-4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2 -b)thiophen-9(10H)-one.
Claim 8
Dependent Claim
9 words
The compound of claim 1, which is 6-chloro-4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2 -b)thiophen-10(9H)-one.
Claim 9
Dependent Claim
9 words
The compound of claim 1, which is 4-(1-isopropyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen -9(20H)-one.
Claim 10
Dependent Claim
8 words
The compound of claim 1, which is 4-(1-n-butyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen-9(10H)-one.
Claim 11
Dependent Claim
9 words
The compound of claim 1, which is 7-chloro-4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2 -b)thiophen-10(9H)-one.
Claim 12
Dependent Claim
9 words
The compound of claim 1, which is 7-chloro-4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2 -b)thiophen-9(10H)-one.
Claim 13
Dependent Claim
8 words
The compound of claim 1, which is 6-bromo-4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen-10(9H)-one.
Claim 14
Dependent Claim
8 words
The compound of claim 1, which is 6-bromo-4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2-b)thiophen-9(10H)-one.
Claim 15
Dependent Claim
9 words
The compound of claim 1, which is 7-methoxy-4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2 -b)thiophen-10(9H)-one.
Claim 16
Dependent Claim
9 words
The compound of claim 1, which is 7-methoxy-4-(1-methyl-4-piperidylidene)-4H-benzo(4,5)cyclohepta(1,2 -b)thiophen-9(10H)-one.
Claim 17
Dependent Claim
5 words
A compound of the formula
Claim 18
Dependent Claim
10 words
A compound of claim 18 in which R2 is methyl.
Claim 19
Dependent Claim
5 words
A compound of the formula:
References Cited (Backward Citations)
US3272826A
Cited
US3491103A
Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1975-08-08 | 1976-02-07 | 1976-08-08 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1979-08-08 | 1980-02-07 | 1980-08-08 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1983-08-08 | 1984-02-07 | 1984-08-08 | $7700.00 | Window Closed / Lapsed |