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US3676447A Expired / Lapsed US ⏱️ 0.0 years remaining

3,4,5-trimethoxybenzamides of phenyl-and pyridylakylamines

Assignee: SRI International Inc
•
Filing: 1970-06-24
•
Granted: 1972-07-11
•
Expires: 1990-06-24
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Abstract

Abstract 3,4,5-Trimethoxybenzamides of pyridylalkylamines such as pyridylmethylamine and of phenylalkylamines such as phenylmethylamine, phenethylamine and Beta hydroxyphenethylamine, as well as derivatives thereof wherein the aromatic nucleus in the amine is substituted by one or more hydroxy, carboxy, halo, aryl, alkyl, nitro, alkoxy, aryloxy or thioalkoxy groups. The compounds are relatively non-toxic and are useful for pharmacological purposes. They exert a specific effect on the central nervous system and a somewhat lesser effect on muscle function. They are useful as relatively mild tranquilizers in the control of anxiety states, excessive aggressiveness and hyperactivity.

Inventors

  • 👤 Wilfred A Skinner
  • 👤 John G Johansson
  • 👤 Howard L Johnson

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-08 06:28
CPC Classifications
C; C07; C07D; C07D213/00; C07D213/02; C07D213/04; C07D213/24; C07D213/36; C07D213/40; C07D213/60; C07D213/62; C07D213/70; C07D213/78; C07D213/81; C07D317/00; C07D317/08; C07D317/44; C07D317/46; C07D317/48; C07D317/50; C07D317/58

Claims Analysis

Total Claims: 21
Claim 1
Independent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(p-ethoxphenyl)- Beta -hydroxyethylamine.
Claim 2
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -hydroxy- Beta -phenethylamine.
Claim 3
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(3,4,5-trimethoxyphenyl)- Beta -hydroxyethylamine.
Claim 4
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(3,4,5biphenylyl)- Beta -hydroxyethylamine.
Claim 5
Dependent Claim 13 words
The compound of claim 1 is the 3,4,5-trimethoxybenzamide of Beta -(p-methoxyphenyl)- Beta -hydroxyethylamine.
Claim 6
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(o-chlorophenyl)- Beta -hydroxyethylamine.
Claim 7
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(m-bromophenyl)- Beta -hydroxyethylamine.
Claim 8
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(3,4-methylenedioxyphenyl)- Beta -hydroxyethylamine.
Claim 9
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(3-fluoro-4-methoxyphenyl)- Beta -hydroxyethylamine.
Claim 10
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(2,6-dichlorophenyl)- Beta -hydroxyethylamine.
Claim 11
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(2,5-dimethoxyphenyl)- Beta -hydroxyethylamine.
Claim 12
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(p-isopropylphenyl)- Beta -hydroxyethylamine.
Claim 13
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(3-methoxy-4-ethoxyphenyl)- Beta -hydroxyethylamine.
Claim 14
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(m-methoxyphenyl)- Beta -hydroxyethylamine.
Claim 15
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(o-methoxyphenyl)- Beta -hydroxyethylamine.
Claim 16
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(2,4-dimethoxyphenyl)- Beta -hydroxyethylamine.
Claim 17
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(0-fluorophenyl- Beta -hydroxyethylamine.
Claim 18
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(2-hydroxy-3-methoxyphenyl)- Beta -hydroxyethylamine.
Claim 19
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(3,4-dibenzyloxyphenyl)- Beta -hydroxyethylamine.
Claim 20
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(o-methylphenyl)- Beta -hydroxyethylamine.
Claim 21
Dependent Claim 14 words
The compound of claim 1 which is the 3,4,5-trimethoxybenzamide of Beta -(o-bromophenyl)- Beta -hydroxyethylamine.

References Cited (Backward Citations)

US2870156A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1975-07-11 1976-01-10 1976-07-11 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1979-07-11 1980-01-10 1980-07-11 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1983-07-11 1984-01-10 1984-07-11 $7700.00 Window Closed / Lapsed

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