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EP0048501A1 Expired / Lapsed EP ⏱️ 0.0 years remaining

Optically active or racemic diazabicyclooctane derivatives

Assignee: Sumitomo Chemical Co Ltd
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Filing: 1979-11-02
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Granted: —
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Expires: 1999-11-02
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Abstract

Abstract Optically active or racemic diazabicyclooctane derivatives of formula wherein A represents a C 6 -C 14 aryl group or a C 1 -C 4 alkyl or alkoxy group- or halogen-substituted C 6 -C 14 aryl group and R 3 represents a C 1 -C 4 alkyl group. These compounds can be prepared by reacting a glyoxylate ester or glyoxylate ester hemiacetal with a 2(-N-substituted aminomethyl)pyrrolidine, and can be used to prepare optically active and racemic α-hydroxyaldehydes which are important intermediates in the preparation of pharmaceuticals and agricultural chemicals.

Inventors

  • 👤 Teruaki Mukaiyama
  • 👤 Yoji Sakito
  • 👤 Masatoshi Asami

Bibliographic Details

Application Number —
Jurisdiction EP
Data Source google_patents
Last Synchronized 2026-10-26 02:41
CPC Classifications
C; C07; C07D; C07D487/00; C07D487/02; C07D487/04; C07C; C07C45/00; C07C45/27; C07C45/56; C07C45/562; C07C47/00; C07C47/20; C07C47/26; C07C47/263; C07C47/27; C07C47/277

Claims Analysis

Total Claims: 9
Claim 1
Independent Claim 47 words
An optically active or racemic diazabicyclooctane derivative of formula wherein A represents a C 6 -C 14 aryl group or a C1 - C4 alkyl or alkoxy group- or halogen-substituted C 6 -C 14 aryl group and R 3 represents a C 1 -C 4 alkyl group.
Claim 2
Dependent Claim 47 words
An optically active or racemic diazabicyclooctane derivative of formula wherein A represents a C 6 -C 14 aryl group or a C1 - C4 alkyl or alkoxy group- or halogen-substituted C 6 -C 14 aryl group and R 3 represents a C 1 -C 4 alkyl group.
Claim 3
Dependent Claim 9 words
An optically active or racemic diazabicyclooctane derivative of formula
Claim 4
Dependent Claim 9 words
An optically active or racemic diazabicyclooctane derivative of formula
Claim 5
Dependent Claim 9 words
An optically active or racemic diazabicyclooctane derivative of formula
Claim 6
Dependent Claim 9 words
An optically active or racemic diazabicyclooctane derivative of formula
Claim 7
Dependent Claim 8 words
An optically active or racemic diazabicyclooctane derivative.of formula
Claim 8
Dependent Claim 8 words
An optically active or racemic diazabicyclooctane derivative.of formula
Claim 9
Dependent Claim 63 words
A process for preparing an optically active or racemic glyoxylic acid derivative of formula wherein A and R 3 are as defined in any one of the preceding claims, which comprises reacting a glyoxylate ester or a glyoxylate ester hemiacetal with an optically active or racemic 2-(N-substituted aminomethyl) pyrrolidine of formula wherein A is as defined in any one of the preceding claims.

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