USRE28939E
Expired / Lapsed
US
⏱️ 0.0 years remaining
3-Aminoindazole derivatives
Assignee: GlaxoSmithKline LLC
•
Filing: 1972-09-28
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Granted: 1976-08-24
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Expires: 1992-09-28
Abstract
Abstract .Iadd.Pharmaceutical compositions having muscle relaxant and analgesic activity containing 3-aminoindazoles..Iaddend.
Inventors
- 👤 John J. Lafferty
- 👤 David H. Tedeschi
- 👤 Charles L. Zirkle
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-07 15:38
CPC Classifications
C; C07; C07D; C07D231/00; C07D231/54; C07D231/56
Claims Analysis
Total Claims: 9
Claim 1
Independent Claim
122 words
A .Iadd.pharmaceutical composition having analgesic and muscle relaxant activity, in dosage unit form, comprising a solid pharmaceutical carrier and from about 25 mg. to about 350 mg. of a .Iaddend.chemical compound of the class consisting of a free base and its nontoxic, pharmaceutically acceptable acid addition salts, the free base having the formula: ##SPC6## in which: R is a member selected from the group consisting of halogen having an atomic weight of less than 80 and trifluoromethyl, said member being in a position β to the hetero ring; R 1 is a member selected from the group consisting of hydrogen, lower alkyl and phenyl; and R 2 and R 3 are members selected from the group consisting of hydrogen and lower alkyl.
Claim 2
Dependent Claim
122 words
A .Iadd.pharmaceutical composition having analgesic and muscle relaxant activity, in dosage unit form, comprising a solid pharmaceutical carrier and from about 25 mg. to about 350 mg. of a .Iaddend.chemical compound of the class consisting of a free base and its nontoxic, pharmaceutically acceptable acid addition salts, the free base having the formula: ##SPC6## in which: R is a member selected from the group consisting of halogen having an atomic weight of less than 80 and trifluoromethyl, said member being in a position β to the hetero ring; R 1 is a member selected from the group consisting of hydrogen, lower alkyl and phenyl; and R 2 and R 3 are members selected from the group consisting of hydrogen and lower alkyl.
Claim 3
Dependent Claim
50 words
A .Iadd.pharmaceutical composition having analgesic and muscle relaxant activity, in dosage unit form, comprising a solid pharmaceutical carrier and from about 25 mg. to about 350 mg. of a .Iaddend.chemical compound of the formula: ##SPC7## in which the CF 3 moiety is in a position β to the hetero ring.
Claim 4
Dependent Claim
50 words
A .Iadd.pharmaceutical composition having analgesic and muscle relaxant activity, in dosage unit form, comprising a solid pharmaceutical carrier and from about 25 mg. to about 350 mg. of a .Iaddend.chemical compound of the formula: ##SPC7## in which the CF 3 moiety is in a position β to the hetero ring.
Claim 5
Dependent Claim
9 words
.Iadd.A pharmaceutical composition of claim 2 containing .Iaddend. 3-amino-5-trifluoromethylindazole.
Claim 6
Dependent Claim
9 words
.Iadd.A pharmaceutical composition of claim 2 containing .Iaddend. 3-amino-6-trifluoromethylindazole.
Claim 7
Dependent Claim
49 words
.Iadd.A pharmaceutical composition having analgesic and muscle relaxant activity, in dosage unit form, comprising a solid pharmaceutical carrier and from about 25 mg. to about 350 mg. of a .Iaddend.chemical compound of the formula: ##SPC8## in which the Cl moiety is in a position β to the hetero ring.
Claim 8
Dependent Claim
49 words
.Iadd.A pharmaceutical composition having analgesic and muscle relaxant activity, in dosage unit form, comprising a solid pharmaceutical carrier and from about 25 mg. to about 350 mg. of a .Iaddend.chemical compound of the formula: ##SPC8## in which the Cl moiety is in a position β to the hetero ring.
Claim 9
Dependent Claim
19 words
.Iadd.A pharmaceutical composition of claim 5 containing .Iaddend. 3-amino-5-chloroindazole. .Iadd.7. A pharmaceutical composition of claim 5 containing .Iaddend. 3-amino-6-chloroindazole.
References Cited (Backward Citations)
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1979-08-24 | 1980-02-23 | 1980-08-24 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1983-08-24 | 1984-02-23 | 1984-08-24 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1987-08-24 | 1988-02-23 | 1988-08-24 | $7700.00 | Window Closed / Lapsed |