US5502233A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Enamine intermediates for the preparation of substituted pyridylpyrimidines
Assignee: Bayer AG
•
Filing: 1995-01-23
•
Granted: 1996-03-26
•
Expires: 2015-01-23
Abstract
Abstract ##STR1## Substituted pyridylpyrimidines have formula (I), in which A and Ar have the meaning given in the test of the description. Also disclosed are their preparation, their use and new initial products. The compounds having formula (I) may be prepared from appropriate salts of 2-pyridylamidine with appropriate enamines; said enamines are also new and disclosed by the invention, and may be prepared from appropriate ketones with appropriate formaldehyde derivates.
Inventors
- 👤 Ulrich Heinemann
- 👤 Heinz-Wilhelm Dehne
- 👤 Stefan Dutzmann
- 👤 Christoph Erdelen
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-09 13:29
CPC Classifications
C; C07; C07D; C07D401/00; C07D401/02; C07D401/04; A; A01; A01N; A01N43/00; A01N43/48; A01N43/54; C07C; C07C225/00; C07C225/02; C07C225/14; C07C225/16; C07C323/00; C07C323/23; C07C323/24; C07C323/27
Claims Analysis
Total Claims: 3
Claim 1
Independent Claim
156 words
An enamine of the formula ##STR307## in which A represents a radical of the formula ##STR308## where R in each case is alkyl X represents oxygen or sulphur and Ar represents phenyl which is optionally monosubstituted to pentasubstituted by identical or different substituents, wherein the substituents are halogen, cyano, nitro, straight-chain or branched alkyl, straight-chain or branched alkoxy or straight-chain or branched alkyl thio, each having 1 to 4 carbon atoms in the alkyl moieties, straight-chain or branched halogenoalkyl, straight-chain or branched halogenoalkoxy or straight-chain or branched halogenoalkylthio, each having 1 to 4 carbon atoms in the alkyl moiety and 1 to 9 identical or different halogen atoms, straight-chain or branched alkoxycarbonyl or alkoxyiminoalkyl, each having 1 to 4 carbon atoms in the individual alkyl moieties, or phenyl which is optionally monosubstituted to pentasubstituted by identical or different substituents from the group consisting of halogen and straight-chain or branched alkyl having 1 to 4 carbon atoms.
Claim 2
Dependent Claim
156 words
An enamine of the formula ##STR307## in which A represents a radical of the formula ##STR308## where R in each case is alkyl X represents oxygen or sulphur and Ar represents phenyl which is optionally monosubstituted to pentasubstituted by identical or different substituents, wherein the substituents are halogen, cyano, nitro, straight-chain or branched alkyl, straight-chain or branched alkoxy or straight-chain or branched alkyl thio, each having 1 to 4 carbon atoms in the alkyl moieties, straight-chain or branched halogenoalkyl, straight-chain or branched halogenoalkoxy or straight-chain or branched halogenoalkylthio, each having 1 to 4 carbon atoms in the alkyl moiety and 1 to 9 identical or different halogen atoms, straight-chain or branched alkoxycarbonyl or alkoxyiminoalkyl, each having 1 to 4 carbon atoms in the individual alkyl moieties, or phenyl which is optionally monosubstituted to pentasubstituted by identical or different substituents from the group consisting of halogen and straight-chain or branched alkyl having 1 to 4 carbon atoms.
Claim 3
Dependent Claim
78 words
An enamine according to claim 1 wherein Ar represents phenyl which is optionally monosubstituted to trisubstituted by identical or different substituents, wherein the substituents are fluorine, chlorine, bromine, cyano, nitro, methyl, ethyl, n-or i-propyl, n-, i-, s-or t-butyl, methoxy, ethoxy, n- or i-propoxy, methylthio, trifluoromethyl, trifluoromethoxy, trifluoromethylthio, methoxycarbonyl, ethoxycarbonyl, methoxyiminomethyl, ethoxyiminomethyl, methoxyiminoethyl, ethoxyiminoethyl, or phenyl which is optionally monosubstituted to trisubstituted by identical or different substituents selected from the group consisting of fluorine, chlorine, bromine, methyl or ethyl.
References Cited (Backward Citations)
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1999-03-26 | 1999-09-25 | 2000-03-26 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 2003-03-26 | 2003-09-25 | 2004-03-26 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 2007-03-26 | 2007-09-25 | 2008-03-26 | $7700.00 | Window Closed / Lapsed |