US4875923A
Expired / Lapsed
US
⏱️ 0.0 years remaining
N-pyridinylsulfonyl-N'-pyrimidinylures
Assignee: Novartis Corp
•
Filing: 1987-10-26
•
Granted: 1989-10-24
•
Expires: 2007-10-26
Abstract
Abstract N-Pyridinylsulfonyl-N'-pyrimidinylureas and N-pyridinylsulfonyl-N'-triazinylureas of the formula ##STR1## wherein E is nitrogen or the methine bridge, Z is oxygen or sulfur, R 4 is hydrogen or C 1 -C 4 alkyl, R 5 and R 6 are each independently hydrogen, halogen, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy, C 1 -C 4 haloalkoxy, C 2 -C 4 -alkylthio, C 3 -C 6 cycloalkyl or --NR 12 R 13 , G is a ##STR2## R 1 is hydrogen, halogen, nitro, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, trifluoromethyl, trifluoromethoxy, difluoromethoxy, C 1 -C 4 alkyl carbonyl or --COOR 14 , R 3 is a ##STR3## group, n is 0, 1 or 2, R 8 is hydrogen, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, halogen, C 1 -C 4 haloalkyl, nitro, --COOR 14 , C 1 -C 4 haloalkoxy, --O--CR 15 R 16 --CN, R 9 is hydrogen, halogen, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 2 -C 4 alkoxyalkyl oder C 2 -C 4 alkoxylkoxy, R 10 and R 11 are each independently hydrogen or C 1 -C 4 alkyl, R 12 and R 13 are each independently hydrogen or C 1 -C 4 alkyl, R 14 is hydrogen, C 1 -C 4 alkyl, C 2 -C 4 alkenyl, C 3 -C 4 alkynyl, or is C 1 -C 4 alkyl which is substituted by C 1 -C 4 alkoxy, halogen or phenyl, and R 15 and R 16 are each independently hydrogen or C 1 -C 4 alkyl, and the salts thereof have useful selective herbicidal properties for controlling weeds in crops of useful plants.
Inventors
- 👤 Rolf Schurter
- 👤 Willy Meyer
- 👤 Werner Fory
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-10-27 11:51
CPC Classifications
C; C07; C07D; C07D333/00; C07D333/50; C07D333/52; C07D333/62; A; A01; A01N; A01N47/00; A01N47/08; A01N47/28; A01N47/36; C07D333/02; C07D333/04; C07D333/26; C07D333/30; C07D333/34; C07D333/38; C07D521/00
Claims Analysis
Total Claims: 15
Claim 1
Independent Claim
288 words
A sulfonylurea of formula I ##STR12## wherein E is the methine bridge, Z is oxygen or sulfur, R 4 is hydrogen or C 1 -C 4 alkyl, R 5 and R 6 are each independently hydrogen, halogen, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy, C 1 -C 4 haloalkoxy, C 1 -C 4 alkylthio, C 3 -C 6 dialkoxyalkyl, C 1 -C 4 haloalkylthio, C 2 -C 4 -alkoxyalkyl, C 3 -C 6 -cycloalkyl or --NR 12 R 13 , G is a ##STR13## R 1 is hydrogen, halogen, nitro, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, trifluoromethyl, trifluoromethoxy, difluoromethoxy, C 1 -C 4 alkyl carbonyl or --COOR 14 , R 3 is a ##STR14## group, n is 0, 1 or 2, R 8 is hydrogen, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, halogen, C 1 -C 4 haloalkyl, nitro, --COOR 14 , C 1 -C 4 haloalkoxy, --O--CR 15 R 16 --COOR 14 or --O--CR 15 R 16 --CN, R 9 is hydrogen, halogen, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 2 -C 4 alkoxyalkyl oder C 2 -C 4 alkoxyalkoxy, R 10 and R 11 are each independently hydrogen or C 1 -C 4 alkyl, R 12 and R 13 are each independently hydrogen or C 1 -C 4 alkyl, R 14 is hydrogen, C 1 -C 4 alkyl, C 2 -C 4 alkenyl, C 3 -C 4 alkynyl, or is C 1 -C 4 alkyl which is substituted by C 1 -C 4 alkoxy, halogen or phenyl, and R 15 and R 16 are each independently hydrogen or C 1 -C 4 alkyl, or a salt thereof.
Claim 2
Dependent Claim
288 words
A sulfonylurea of formula I ##STR12## wherein E is the methine bridge, Z is oxygen or sulfur, R 4 is hydrogen or C 1 -C 4 alkyl, R 5 and R 6 are each independently hydrogen, halogen, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy, C 1 -C 4 haloalkoxy, C 1 -C 4 alkylthio, C 3 -C 6 dialkoxyalkyl, C 1 -C 4 haloalkylthio, C 2 -C 4 -alkoxyalkyl, C 3 -C 6 -cycloalkyl or --NR 12 R 13 , G is a ##STR13## R 1 is hydrogen, halogen, nitro, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, trifluoromethyl, trifluoromethoxy, difluoromethoxy, C 1 -C 4 alkyl carbonyl or --COOR 14 , R 3 is a ##STR14## group, n is 0, 1 or 2, R 8 is hydrogen, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, halogen, C 1 -C 4 haloalkyl, nitro, --COOR 14 , C 1 -C 4 haloalkoxy, --O--CR 15 R 16 --COOR 14 or --O--CR 15 R 16 --CN, R 9 is hydrogen, halogen, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 2 -C 4 alkoxyalkyl oder C 2 -C 4 alkoxyalkoxy, R 10 and R 11 are each independently hydrogen or C 1 -C 4 alkyl, R 12 and R 13 are each independently hydrogen or C 1 -C 4 alkyl, R 14 is hydrogen, C 1 -C 4 alkyl, C 2 -C 4 alkenyl, C 3 -C 4 alkynyl, or is C 1 -C 4 alkyl which is substituted by C 1 -C 4 alkoxy, halogen or phenyl, and R 15 and R 16 are each independently hydrogen or C 1 -C 4 alkyl, or a salt thereof.
Claim 3
Dependent Claim
10 words
A compound according to claim 1, wherein Z is oxygen.
Claim 4
Dependent Claim
30 words
A compound according to claim 1, wherein R 1 is hydrogen, Cl, F, CH 3 , C 2 H 5 , CH 3 O, CF 3 or CH 3 CO.
Claim 5
Dependent Claim
25 words
A compound according to claim 1, wherein R 5 and R 6 together contain not more than 4 carbon atoms and R 4 is hydrogen.
Claim 6
Dependent Claim
10 words
A compound according to claim 1, wherein G is 3-phenylpyridin-2-yl.
Claim 7
Dependent Claim
32 words
A compound according to claim 1, wherein Z is oxygen, R 4 is hydrogen and G is 3-phenylpyridin-2-yl and R 5 and R 6 together contain not more than 4 carbon atoms.
Claim 8
Dependent Claim
5 words
N-(3-Phenylpyridin-2-ylsulfonyl)-N'-(4,6-dimethoxypyrimidin-2-yl)urea according to claim 1.
Claim 9
Dependent Claim
30 words
A herbicidal and plant growth inhibiting composition which contains, as active ingredient, at least one substituted sulfonylurea of formula I according to claim 1, together with carriers and/or other adjuvants.
Claim 10
Dependent Claim
40 words
A method of controlling undesired plant growth, which method comprises applying to the plants or to the locus thereof an effective amount of a compound of formula I according to claim 1, or of a composition containing such a compound.
Claim 11
Dependent Claim
39 words
A method of inhibiting plant growth, which method comprises applying to the plants or to the locus thereof an effective amount of a compound of formula I according to claim 1, or of a composition containing such a compound.
Claim 12
Dependent Claim
42 words
A method of influencing plant growth for increasing yield, which method comprises applying to the plants or to the locus thereof an effective amount of a compound of formula I according to claim 1, or of a composition containing such a compound.
Claim 13
Dependent Claim
18 words
A method according to claim 9 of selectively controlling weeds pre- or postemergence in crops of useful plants.
Claim 14
Dependent Claim
22 words
A method according to claim 10 of suppressing plant growth beyond the 2-leaf stage, which method comprises applying the active ingredient preemergence.
Claim 15
Dependent Claim
12 words
A method according to claim 12, wherein the crops are rice crops.
References Cited (Backward Citations)
CH580608A5
Cited
DE3105453A1
Cited
EP0071441A2
Cited
EP0096593A2
Cited
DE3225471A1
Cited
US4668279A
Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1992-10-23 | 1993-04-24 | 1993-10-24 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1996-10-23 | 1997-04-24 | 1997-10-24 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 2000-10-23 | 2001-04-24 | 2001-10-24 | $7700.00 | Window Closed / Lapsed |