Claims Analysis
Total Claims: 14
Claim 1
Independent Claim
453 words
A 5-acylamino-pyrazole derivative of the formula ##STR193## in which R 1 represents hydrogen, nitro, flourine, chlorine, bromine or iodine; R 2 represents hydrogen, or represents straight-chain or branched alkyl with 1 to 12 carbon atoms, or represents in each case straight-chain or branched alkenyl or alkinyl with in each case 3 to 8 carbon atoms, or represents cycloalkyl which has 3 to 8 carbon atoms and is optionally substituted by alkyl with 1 to 4 carbon atoms; Ar represents phenyl, 2-pyridyl, 3-pyridyl or 4-pyridyl, in each case optionally substituted by substituents independently selected from the group consisting of halogen, cyano, nitro, in each case straight-chain or branched alkyl, alkoxy and alkoxycarbonyl with in each case 1 to 4 carbon atoms in the alkyl parts, in each case straight-chain or branched halogenoalkyl and halogenoalkoxy with in each case 1 to 4 carbon atoms and 1 to 9 identical or different halogen atoms and an --S(O) m --R 4 radical, wherein R 4 represents amino, or represents in each case straight-chain or branched alkyl, alkylamino, dialkylamino or halogenoalkyl with in each case 1 to 4 carbon atoms in the individual alkyl parts and in the case of the halogenoalkyl with 1 to 9 identical or different halogen atoms and m represents the number 0, 1 or 2; and X represents oxygen or sulphur; A represents a straight-chain or branched alkylene bridge which has 1 to 6 carbon atoms and is optionally monosubstituted or polysubstituted by identical or different substituents from the group comprising halogen and phenyl, which is optionally substituted by halogen or alkyl with 1 to 4 carbon atoms; n represents the number 0 or 1 and Y represents cyano or the grouping ##STR194## wherein X 1 represents oxygen or sulphur and R 3 represents hydroxyl, in each case straight-chain or branched alkoxy or alkylthio with in each case 1 to 6 carbon atoms, in each case straight-chain or branched alkenyloxy or alkinyloxy with in each case 3 to 8 carbon atoms, amino, in each case straight-chain or branched alkylamino or dialkylamino with in each case 1 to 6 carbon atoms in the alkyl parts, in each case straight-chain or branched alkenylamino or dialkenylamino with in each case 3 to 8 carbon atoms in the alkenyl parts or straight-chain or branched alkyl-alkenylamino with 1 to 6 carbon atoms in the alkyl part and 3 to 8 carbon atoms in the alkenyl part, or represents an --OM radical, wherein M represents one equivalent of an alkaline earth metal cation or alkali metal cation, or represents ammonium which is optionally mono-, di-, tri- or tetrasubstituted by identical or different substituents from the group comprising straight-chain or branched alkyl with 1 to 12 carbon atoms and benzyl.
Claim 2
Dependent Claim
453 words
A 5-acylamino-pyrazole derivative of the formula ##STR193## in which R 1 represents hydrogen, nitro, flourine, chlorine, bromine or iodine; R 2 represents hydrogen, or represents straight-chain or branched alkyl with 1 to 12 carbon atoms, or represents in each case straight-chain or branched alkenyl or alkinyl with in each case 3 to 8 carbon atoms, or represents cycloalkyl which has 3 to 8 carbon atoms and is optionally substituted by alkyl with 1 to 4 carbon atoms; Ar represents phenyl, 2-pyridyl, 3-pyridyl or 4-pyridyl, in each case optionally substituted by substituents independently selected from the group consisting of halogen, cyano, nitro, in each case straight-chain or branched alkyl, alkoxy and alkoxycarbonyl with in each case 1 to 4 carbon atoms in the alkyl parts, in each case straight-chain or branched halogenoalkyl and halogenoalkoxy with in each case 1 to 4 carbon atoms and 1 to 9 identical or different halogen atoms and an --S(O) m --R 4 radical, wherein R 4 represents amino, or represents in each case straight-chain or branched alkyl, alkylamino, dialkylamino or halogenoalkyl with in each case 1 to 4 carbon atoms in the individual alkyl parts and in the case of the halogenoalkyl with 1 to 9 identical or different halogen atoms and m represents the number 0, 1 or 2; and X represents oxygen or sulphur; A represents a straight-chain or branched alkylene bridge which has 1 to 6 carbon atoms and is optionally monosubstituted or polysubstituted by identical or different substituents from the group comprising halogen and phenyl, which is optionally substituted by halogen or alkyl with 1 to 4 carbon atoms; n represents the number 0 or 1 and Y represents cyano or the grouping ##STR194## wherein X 1 represents oxygen or sulphur and R 3 represents hydroxyl, in each case straight-chain or branched alkoxy or alkylthio with in each case 1 to 6 carbon atoms, in each case straight-chain or branched alkenyloxy or alkinyloxy with in each case 3 to 8 carbon atoms, amino, in each case straight-chain or branched alkylamino or dialkylamino with in each case 1 to 6 carbon atoms in the alkyl parts, in each case straight-chain or branched alkenylamino or dialkenylamino with in each case 3 to 8 carbon atoms in the alkenyl parts or straight-chain or branched alkyl-alkenylamino with 1 to 6 carbon atoms in the alkyl part and 3 to 8 carbon atoms in the alkenyl part, or represents an --OM radical, wherein M represents one equivalent of an alkaline earth metal cation or alkali metal cation, or represents ammonium which is optionally mono-, di-, tri- or tetrasubstituted by identical or different substituents from the group comprising straight-chain or branched alkyl with 1 to 12 carbon atoms and benzyl.
Claim 3
Dependent Claim
339 words
A 5-acylamino-pyrazole derivative according to claim 1, in which R 1 represents hydrogen, nitro, chlorine or bromine, R 2 represents hydrogen, or represents straight-chain or branched alkyl with 1 to 8 carbon atoms, or represents in each case straight-chain or branched alkenyl or alkinyl with in each case 3 to 6 carbon atoms, or represents cycloalkyl which has 3 to 6 carbon atoms and is optionally substituted by methyl, ethyl or isopropyl; Ar represents phenyl which is optionally mono-, di-, tri-, tetra- or pentasubstituted by identical or different substituents, or represents 2-pyridyl, 3-pyridyl or 4-pyridyl, in each case optionally mono-, di-, tri- or tetrasubstituted by identical or different substituents, the substituents in each case being cyano, nitro, fluorine, chlorine, bromine, iodine, methyl, ethyl, n- and i-propyl, n-, i-, s- and t-butyl, methoxy, ethoxy, methoxycarbonyl, ethoxycarbonyl, trifluoromethyl, trichloromethyl, dichlorofluoromethyl, difluorochloromethyl, chloromethyl, dichloromethyl, difluoromethyl, pentafluoroethyl, tetrafluoroethyl, trifluorochloroethyl, trifluoroethyl, difluorodichloroethyl, trifluorodichloroethyl, pentachloroethyl, trifluoromethoxy, trichloromethoxy, dichlorofluoromethoxy, difluorochloromethoxy, chloromethoxy, dichloromethoxy) difluoromethoxy, pentafluoroethoxy, tetrafluoroethoxy, trifluorochloroethoxy, trifluoroethoxy, difluorodichloroethoxy, trifluorodichloroethoxy, pentachloroethoxy or an --S(O) m --R 4 radical, wherein R 4 represents amino, methylamino, ethylamino, dimethylamino, diethylamino, fluorodichloromethyl, difluoromethyl, tetrafluoroethyl, trichloroethyl, trifluoromethyl, difluorochloromethyl, methyl or ethyl and m represents the number 0, 1 or 2, and X represents oxygen or sulphur; A represents a bridge member of the formula ##STR195## n represents the number 0 or 1 and Y represents cyano or the grouping ##STR196## wherein X 1 represents oxygen and R 3 represents hydroxyl, alkoxy with 1 to 3 carbon atoms, alkenyloxy or alkinyloxy with in each case 3 to 6 carbon atoms, amino, alkylamino or dialkylamino with in each case 1 to 3 carbon atoms in each alkyl part, alkenylamino or dialkenylamino with in each case 3 to 6 carbon atoms in each alkenyl part or alkyl-alkenylamino with 1 to 3 carbon atoms in the alkyl part and 3 to 6 carbon atoms in the alkenyl part, or represents an --OM radical, wherein M represents one equivalent of a sodium, potassium, calcium, magnesium or barium cation, or represents an isopropylammonium, dimethylbenzylammonium, triethylammonium or tributylammonium ion.
Claim 4
Dependent Claim
15 words
A compound according to claim 1, wherein such compound is 5-cyanoacetylamino-1-(2,6-dichloro-4-trifluoromethyl-phenyl)-4-nitro-pyrazole of the formula ##STR197##
Claim 5
Dependent Claim
15 words
A compound according to claim 1, wherein such compound is 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(ethoxycarbonyl-acetamido)-4nitro-pyrazole of the formula ##STR198##
Claim 6
Dependent Claim
15 words
A compound according to claim 1, wherein such compound is 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(1-ethoxycarbonyl-propionylamido)-4-nitro-pyrazole of the formula ##STR199##
Claim 7
Dependent Claim
15 words
A compound according to claim 1, wherein such compound is 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(ethoxalylamido)-4-nitro-pyrazole of the formula ##STR200##
Claim 8
Dependent Claim
15 words
A compound according to claim 1, wherein such compound is 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(sodiooxalylamido)-4-nitro-pyrazole of the formula ##STR201##
Claim 9
Dependent Claim
18 words
A herbicidal composition comprising a herbicidally effective amount of a compound according to claim 1 and a diluent.
Claim 10
Dependent Claim
36 words
A method of killing unwanted vegetation which comprises applying to such vegetation or to a locus from which it is desired to exclude such vegetation a herbicidally effective amount of a compound according to claim 1.
Claim 11
Dependent Claim
16 words
The method according to claim 9, wherein such compound is 5-cyanoacetylamino-1-(2,6-dichloro-4-trifluoromethyl-phenyl)-4-nitro-pyrazole, 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(ethoxycarbonyl-acetamido)-4-nitro-pyrazole, 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(1-ethoxycarbonyl-propionylamido)-4-nitro-pyrazole, 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(ethoxalylamido)-4-nitro-pyrazole, or 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(sodiooxalylamido)-4-nitro-pyrazole.
Claim 12
Dependent Claim
19 words
A plant growth-regulating compositon comprising a plant-growth-regulating effective amount of a compound according to claim 1 and a diluent.
Claim 13
Dependent Claim
41 words
A method of regulating the growth of plants which comprises applying to such plants or to a locus in which such plants are growing or are to be grown a plant growth-regulating effective amount of a compound according to claim 1.
Claim 14
Dependent Claim
16 words
The method according to claim 12, wherein such compound is 5-cyanoacetylamino-1-(2,6-dichloro-4-trifluoromethyl-phenyl)-4-nitro-pyrazole, 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(ethoxycarbonyl-acetamido)-4-nitro-pyrazole, 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(1-ethoxycarbonyl-propionylamido)-4-nitro-pyrazole, 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(ethoxalylamido)-4-nitro-pyrazole, or 1-(2,6-dichloro-4-trifluoromethyl-phenyl)-5-(sodiooxalylamido)-4-nitro-pyrazole.