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US4546113A Expired / Lapsed US ⏱️ 0.0 years remaining

Antiprotozoal diamidines

Assignee: Pfizer Inc
•
Filing: 1983-04-14
•
Granted: 1985-10-08
•
Expires: 2003-04-14
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Abstract

Abstract Diamidines of the formula ##STR1## wherein X is a propylene, isobutylene, guanidine, pyrrole, tetrazole, imidazole or substituted imidazole group; and 2-[4-(2-imidazolinyl)phenyl]-6-(2-imidazolinyl)indole, are useful in the treatment of certain protozoal infections in mammals, particularly in cattle.

Inventors

  • 👤 Edward A. Glazer

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-06 12:20
CPC Classifications
C; C07; C07D; C07D207/00; C07D207/02; C07D207/30; C07D207/32; C07D207/33; C07D207/337; C07C; C07C255/00; C07D233/00; C07D233/54; C07D233/64; C07D257/00; C07D257/02; C07D257/04; C07D401/00; C07D401/02; C07D401/12

Claims Analysis

Total Claims: 6
Claim 1
Independent Claim 18 words
A compound of the formula ##STR20## wherein X is --CH 2 CH═CH-- or --CH 2 C(CH 3 )═CH--.
Claim 2
Dependent Claim 18 words
A compound of the formula ##STR20## wherein X is --CH 2 CH═CH-- or --CH 2 C(CH 3 )═CH--.
Claim 3
Dependent Claim 11 words
The compound of claim 1 wherein X is --CH 2 CH═CH--.
Claim 4
Dependent Claim 13 words
The compound of claim 1 wherein X is --CH 2 C(CH 3 )═CH--.
Claim 5
Dependent Claim 35 words
A pharmaceutical composition suitable for parenteral administration in the treatment of a protozoal infection in a mammal which comprises an antiprotozoal effective amount of a compound of claim 1 and a pharmaceutically acceptable liquid vehicle.
Claim 6
Dependent Claim 31 words
A method of treating a susceptible protozoal infection in a mammal which comprises parenteral administration of an antiprotozoal effective amount of compound of claim 1 in a pharmaceutically acceptable liquid vehicle.

References Cited (Backward Citations)

US2204983A Cited
GB549634A Cited
US3652591A Cited
US3689506A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1988-10-07 1989-04-08 1989-10-08 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1992-10-07 1993-04-08 1993-10-08 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1996-10-07 1997-04-08 1997-10-08 $7700.00 Window Closed / Lapsed

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