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US4500715A Expired / Lapsed US ⏱️ 0.0 years remaining

2,5-Diamino-1,3,4-thiadiazole derivatives

Assignee: Bayer AG
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Filing: 1981-01-26
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Granted: 1985-02-19
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Expires: 2001-01-26
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Abstract

Abstract 1,3,4-Thiazole derivatives of the formula ##STR1## wherein R 26 ' denotes a C 1 -C 8 -alkyl radical which is optionally substituted by hydroxyl, halogen, cyano, C 1 -C 4 -alkoxy, carboxyl, aminocarbonyl or C 1 -C 4 -alkoxycarbonyl, a C 2 -C 4 -alkenyl radical, a cyclohexyl radical which is optionally substituted by C 1 -C 4 -alkyl, a phenyl, benzyl or phenylethyl radical which is optionally substituted by halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy, a C 1 -C 2 -alkylcarbonyl, C 1 -C 4 -alkoxycarbonyl, mono- or di-C 1 -C 4 -alkylaminocarbonyl, aminocarbonyl, mono- or di-C 1 -C 4 -alkylaminosulphonyl, 2-thienyl, 2-furyl, 2-tetrahydrofuryl, amino, C 1 -C 4 -alkylamino or di-(C 1 -C 4 -alkyl)-amino radical or a phenylamino or benzylamino radical which is optionally substituted by C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy and R 27 ' denotes a C 1 -C 8 -alkyl radical which is optionally substituted by hydroxyl, halogen, cyano, C 1 -C 4 -alkoxy, carboxyl, aminocarbonyl- or C 1 -C 4 -alkoxycarbonyl, a C 2 -C.sub. 4 -alkenyl radical or a benzyl or phenylethyl radical which is substituted by halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy, are useful as intermediates for the preparation of pharmaceuticals, agents for protecting plants and dyestuffs.

Inventors

  • 👤 Hauke Furstenwerth

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-02 11:25
CPC Classifications
C; C07; C07D; C07D285/00; C07D285/01; C07D285/02; C07D285/04; C07D285/12; C07D285/125; C07D285/135; C09; C09B; C09B44/00; C09B44/10; C09B44/107

Claims Analysis

Total Claims: 2
Claim 1
Independent Claim 209 words
Thiadiazole derivatives of the general formula ##STR548## wherein R 26 ' denotes a C 1 -C 8 -alkyl radical which is optionally substituted by hydroxyl, halogen, cyano, C 1 -C 4 -alkoxy, carboxyl, aminocarbonyl or C 1 -C 4 -alkoxycarbonyl, a C 2 -C 4 -alkenyl radical, a cyclohexyl radical which is optionally substituted by C 1 -C 4 -alkyl, a phenyl, benzyl or phenylethyl radical which is optionally substituted by halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy, a C 1 -C 2 -alkylcarbonyl, C 1 -C 4 -alkoxycarbonyl, mono- or di-C 1 -C 4 -alkylaminocarbonyl, aminocarbonyl, mono- or di-C 1 -C 4 -alkylaminosulphonyl, 2-thienyl, 2-furyl, 2-tetrahydrofuryl, amino, C 1 -C 4 -alkylamino or di-(C 1 -C 4 -alkyl)-amino radical or a phenylamino or benzylamino radical which is optionally substituted by C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy and R 27 ' denotes a C 1 -C 8 -alkyl radical which is optionally substituted by hydroxyl, halogen, cyano, C 1 -C 4 -alkoxy, carboxyl, aminocarbonyl- or C 1 -C 4 -alkoxycarbonyl, a C 2 -C 4 -alkenyl radical or a benzyl or phenylethyl radical which is substituted by halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy.
Claim 2
Dependent Claim 209 words
Thiadiazole derivatives of the general formula ##STR548## wherein R 26 ' denotes a C 1 -C 8 -alkyl radical which is optionally substituted by hydroxyl, halogen, cyano, C 1 -C 4 -alkoxy, carboxyl, aminocarbonyl or C 1 -C 4 -alkoxycarbonyl, a C 2 -C 4 -alkenyl radical, a cyclohexyl radical which is optionally substituted by C 1 -C 4 -alkyl, a phenyl, benzyl or phenylethyl radical which is optionally substituted by halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy, a C 1 -C 2 -alkylcarbonyl, C 1 -C 4 -alkoxycarbonyl, mono- or di-C 1 -C 4 -alkylaminocarbonyl, aminocarbonyl, mono- or di-C 1 -C 4 -alkylaminosulphonyl, 2-thienyl, 2-furyl, 2-tetrahydrofuryl, amino, C 1 -C 4 -alkylamino or di-(C 1 -C 4 -alkyl)-amino radical or a phenylamino or benzylamino radical which is optionally substituted by C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy and R 27 ' denotes a C 1 -C 8 -alkyl radical which is optionally substituted by hydroxyl, halogen, cyano, C 1 -C 4 -alkoxy, carboxyl, aminocarbonyl- or C 1 -C 4 -alkoxycarbonyl, a C 2 -C 4 -alkenyl radical or a benzyl or phenylethyl radical which is substituted by halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy.

References Cited (Backward Citations)

US2708671A Cited
FR1199411A Cited
US3096320A Cited
US3639385A Cited
US4006127A Cited
US4036826A Cited
US4082740A Cited
US4281120A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1988-02-19 1988-08-20 1989-02-19 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1992-02-19 1992-08-20 1993-02-19 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1996-02-19 1996-08-20 1997-02-19 $7700.00 Window Closed / Lapsed

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