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US4451282A Expired / Lapsed US ⏱️ 0.0 years remaining

Herbicidally active novel hetero-substituted pyrid-4-one derivatives

Assignee: Bayer AG
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Filing: 1982-08-26
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Granted: 1984-05-29
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Expires: 2002-08-26
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Abstract

Abstract Hetero-substituted pyrid-4-one derivatives of the general formula ##STR1## in which R 1 represents an optionally substituted phenyl radical, R 2 represents an alkyl, alkenyl, alkinyl, alkoxy, alkoxyalkyl or dialkylamino radical, and R 3 and R 4 , together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical, are novel, are produced as described and find use as herbicides, especially as selective herbicides for combating graminaceous weeds in crops such as cotton, wheat, soy beans and corn.

Inventors

  • 👤 Hans-Joachim Knops
  • 👤 Peter Babczinski
  • 👤 Ludwig Eue
  • 👤 Robert Schmidt

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-08 20:22
CPC Classifications
C; C07; C07D; C07D231/00; C07D231/02; C07D231/10; C07D231/12; A; A01; A01N; A01N43/00; A01N43/34; A01N43/40; A01N43/48; A01N43/50; A01N43/56; A01N43/64; A01N43/647; A01N43/653; C07D233/00; C07D233/54; C07D233/56; C07D249/00; C07D249/02; C07D249/08; C07D401/00; C07D401/02; C07D401/04

Claims Analysis

Total Claims: 10
Claim 1
Independent Claim 149 words
A hetero-substituted pyrid-4-one derivative of the formula ##STR32## in which R 1 represents a phenyl radical which is optionally monosubstituted or polysubstituted by identical or different substituents selected from halogen, alkyl, alkoxy or alkylthio, each having 1 to 4 carbon atoms, and halogenoalkyl having 1 or 2 carbon atoms and 1 to 5 identical or different halogen atoms, R 2 represents an alkyl having 1 to 4 carbon atoms, an alkenyl or alkinyl radical, each having 3 to 4 carbon atoms, an alkoxy or alkoxyalkyl radical, each having 1 to 4 carbon atoms in each alkyl part, or a dialkylamino radical having 1 to 4 carbon atoms in each alkyl part, and R 3 and R 4 , together with the nitrogen atom to which they are bonded, represent a heterocyclic radical which is optionally substituted by methyl, methoxy or chlorine and is selected from 1,2,4-triazolyl, imidazolyl and pyrazolyl.
Claim 2
Dependent Claim 149 words
A hetero-substituted pyrid-4-one derivative of the formula ##STR32## in which R 1 represents a phenyl radical which is optionally monosubstituted or polysubstituted by identical or different substituents selected from halogen, alkyl, alkoxy or alkylthio, each having 1 to 4 carbon atoms, and halogenoalkyl having 1 or 2 carbon atoms and 1 to 5 identical or different halogen atoms, R 2 represents an alkyl having 1 to 4 carbon atoms, an alkenyl or alkinyl radical, each having 3 to 4 carbon atoms, an alkoxy or alkoxyalkyl radical, each having 1 to 4 carbon atoms in each alkyl part, or a dialkylamino radical having 1 to 4 carbon atoms in each alkyl part, and R 3 and R 4 , together with the nitrogen atom to which they are bonded, represent a heterocyclic radical which is optionally substituted by methyl, methoxy or chlorine and is selected from 1,2,4-triazolyl, imidazolyl and pyrazolyl.
Claim 3
Dependent Claim 59 words
A compound according to claim 1, in which R 1 represents a phenyl radical which is optionally monosubstituted or disubstituted by identical or different substituents selected from fluorine, chlorine, bromine, methyl, ethyl, isopropyl, methoxy, ethoxy, isopropoxy, methylthio, ethylthio, isopropylthio and trifluoromethyl; and R 2 represents a methyl, ethyl, i-propyl, allyl, propargyl, methoxy, ethoxy, methoxymethyl, ethoxymethyl, ethoxyethyl or dimethylamino radical.
Claim 4
Dependent Claim 15 words
A compound according to claim 1, wherein such compound is 1-methyl-3-(1,2,4-triazol-1-yl)-5-(3-trifluoromethylphenyl)-pyrid-4-one of the formula ##STR33##
Claim 5
Dependent Claim 15 words
A compound according to claim 1, wherein such compound is 1-methyl-3-(pyrazol-1-yl)-5-(3-trifluoromethyl-phenyl)-pyrid-4-one of the formula ##STR34##
Claim 6
Dependent Claim 20 words
A herbicidal composition comprising a herbicidally effective amount of a compound according to claim 1, in admixture with a diluent.
Claim 7
Dependent Claim 21 words
A composition according to claim 5, characterized in that it contains from 0.1 to 95% of the active compound, by weight.
Claim 8
Dependent Claim 26 words
A method of combating weeds, comprising applying to the weeds, or to a habitat thereof, a herbicidally effective amount of a compound according to claim 1.
Claim 9
Dependent Claim 44 words
A method of combating weeds in the growing of a cotton, wheat, soy bean or corn crop comprising applying to the weeds or to the field in which the crop is being grown a herbicidally effective amount of a compound according to claim 3.
Claim 10
Dependent Claim 44 words
A method of combating weeds in the growing of a cotton, wheat, soy bean or corn crop comprising applying to the weeds or to the field in which the crop is being grown a herbicidally effective amount of a compound according to claim 4.

References Cited (Backward Citations)

US4152136A Cited
US4235619A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1987-05-29 1987-11-28 1988-05-29 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1991-05-29 1991-11-28 1992-05-29 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1995-05-29 1995-11-28 1996-05-29 $7700.00 Window Closed / Lapsed

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