US4402953A
Expired / Lapsed
US
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Fungicidal N-(morpholinoacetyl)-anilines, compositions and use
Assignee: Novartis Corp
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Filing: 1980-11-10
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Granted: 1983-09-06
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Expires: 2000-11-10
Abstract
Abstract Amino aceto anilides of the formula I shown hereinafter are effective microbicides. They may be used to control fungi on plants or parts of plants or to prevent them from fungi attack.
Inventors
- 👤 Adolf Hubele
- 👤 Walter Kunz
- 👤 Wolfgang Eckhardt
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-10-27 07:22
CPC Classifications
C; C07; C07D; C07D203/00; C07D203/04; C07D203/06; C07D203/08; A; A01; A01N; A01N37/00; A01N37/44; A01N37/46; C07D207/00; C07D207/02; C07D207/30; C07D207/32; C07D207/325; C07D207/327; C07D211/00; C07D211/04; C07D211/06; C07D211/36; C07D211/38; C07D231/00; C07D231/02; C07D231/10; C07D231/12; C07D233/00; C07D233/54; C07D233/56; C07D249/00; C07D249/02; C07D249/08; C07D295/00; C07D295/04; C07D295/14; C07D295/145; C07D295/15
Claims Analysis
Total Claims: 9
Claim 1
Independent Claim
173 words
A compound of the formula ##STR69## wherein R 1 represents a C 1 -C 4 -alkyl group, a C 1 -C 4 -alkoxy group or a halogen atom, R 2 represents a hydrogen atom, a C 1 -C 3 -alkyl group, a C 1 -C 4 -alkoxy group or a halogen atom, R 3 represents a hydrogen atom, a C 1 -C 3 -alkyl group or a halogen atom, R 4 represents a hydrogen atom or a methyl group, with the proviso that the total number of carbon atoms contained by the substituents R 1 , R 2 , R 3 and R 4 in the phenyl ring does not exceed 8, and X represents --CH 2 -- or ##STR70## R 5 represents --COOR', --COSR' or ##STR71## wherein each of R', R" and R'" independently represents a methyl or ethyl group, R 6 and R 7 together with the nitrogen atom to which they are attached represent morpholine, or salts of the compounds of the formula I with an inorganic or organic acid.
Claim 2
Dependent Claim
173 words
A compound of the formula ##STR69## wherein R 1 represents a C 1 -C 4 -alkyl group, a C 1 -C 4 -alkoxy group or a halogen atom, R 2 represents a hydrogen atom, a C 1 -C 3 -alkyl group, a C 1 -C 4 -alkoxy group or a halogen atom, R 3 represents a hydrogen atom, a C 1 -C 3 -alkyl group or a halogen atom, R 4 represents a hydrogen atom or a methyl group, with the proviso that the total number of carbon atoms contained by the substituents R 1 , R 2 , R 3 and R 4 in the phenyl ring does not exceed 8, and X represents --CH 2 -- or ##STR70## R 5 represents --COOR', --COSR' or ##STR71## wherein each of R', R" and R'" independently represents a methyl or ethyl group, R 6 and R 7 together with the nitrogen atom to which they are attached represent morpholine, or salts of the compounds of the formula I with an inorganic or organic acid.
Claim 3
Dependent Claim
50 words
A compound of the formula I according to claim 1, wherein R 1 represents a methyl group, R 2 is in ortho-position to the amino group and represents a methyl or ethyl group or a chlorine atom, and --X--R 5 represents the group --CH(CH 3 )--COOR' or --CH(CH 3 )--CO--S--R'.
Claim 4
Dependent Claim
79 words
Compounds of the formula I according to claim 1, wherein R 1 represents a methyl or methoxy group, R 2 is in ortho-position to the amino group and represents a methyl or ethyl group, a chlorine or bromine atom, R 3 represents a hydrogen atom, a methyl group, a chlorine or bromine atom, R 4 represents a hydrogen atom or a methyl group, and --X--R 5 represents the group --CH(CH 3 )--COOCH 3 or --CH(CH 3 )--COSCH 3 .
Claim 5
Dependent Claim
9 words
The compound according to claim 3 which is N-(1'-methoxycarbonyl-ethyl)-N-morpholinoacetyl-2,6-dimethylaniline.
Claim 6
Dependent Claim
29 words
A fungicidal composition which contains as active component a fungicidally effective amount of of compound of the formula I according to claim 1, together with a suitable carrier therefor.
Claim 7
Dependent Claim
38 words
A method of controlling phytopathogenic fungi or of preventing fungus attack, which comprises applying to the plants, parts of plants or their environment, a fungicidally effective amount of a compound of the formula I according to claim 1.
Claim 8
Dependent Claim
33 words
A method of controlling phytophathogenic fungi or of preventing fungus attack, which comprises applying to plants, parts of plants or their environment, a fungicidally effective amount of a compound according to claim 3.
Claim 9
Dependent Claim
33 words
A method of controlling phytophathogenic fungi or of preventing fungus attack, which comprises applying to plants, parts of plants or their environment, a fungicidally effective amount of the compound according to claim 4.
References Cited (Backward Citations)
US3108997A
Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1986-09-05 | 1987-03-07 | 1987-09-06 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1990-09-05 | 1991-03-07 | 1991-09-06 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1994-09-05 | 1995-03-07 | 1995-09-06 | $7700.00 | Window Closed / Lapsed |