US4241058A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Heterocyclics useful as fungicides and fungicidal compositions thereof
Assignee: Hoffmann La Roche Inc
•
Filing: 1977-11-18
•
Granted: 1980-12-23
•
Expires: 1997-11-18
Abstract
Abstract Heterocyclic compounds characterized by the formula <IMAGE> I wherein R1, R3, R4, R5, R6, X and z are as hereinafter set forth, prepared, inter alia, by reacting a compound characterized by the formula <IMAGE> II with an amine characterized by the formula <IMAGE> III wherein R1, R3, R4, R5, R6, X and Y are as hereinafter set forth, are described. The end products are useful as fungicidal agents.
Inventors
- 👤 Albert Pfiffner
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-07 17:44
CPC Classifications
C; C07; C07D; C07D295/00; C07D295/02; C07D295/027; C07D295/03; A; A01; A01N; A01N33/00; A01N33/02; A01N33/04; A01N33/16; A01N43/00; A01N43/34; A01N43/40; A01N43/72; A01N43/84; A01N49/00; A61; A61P; A61P17/00; A61P31/00; A61P31/04; C07C; C07C17/00; C07C17/093; C07C17/16; C07C29/00; C07C29/132; C07C29/136; C07C29/14; C07C29/36; C07C29/38; C07C29/40; C07C45/00; C07C45/41; C07C45/51; C07C45/54; C07C45/61; C07C45/62; C07C45/67; C07C45/68; C07C45/72; C07C45/74; C07C47/00; C07C47/20; C07C47/228; C07C47/23; C07C47/232; C07C47/235; C07C49/00; C07C49/20; C07C49/213; C07C49/217; C07D215/00; C07D215/02; C07D215/04; C07D215/06; C07D217/00; C07D217/02; C07D217/04; C07D295/22; C07D295/24
Claims Analysis
Total Claims: 185
Claim 1
Independent Claim
102 words
A compound of the formula ##STR18## , wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; X is a methylene or an oxygen atom; z is zero or 1; and the dotted bonds can be hydrogenated, or an acid addition salt of a compound thereof which is basic.
Claim 2
Dependent Claim
102 words
A compound of the formula ##STR18## , wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; X is a methylene or an oxygen atom; z is zero or 1; and the dotted bonds can be hydrogenated, or an acid addition salt of a compound thereof which is basic.
Claim 3
Dependent Claim
97 words
A compound of the formula ##STR19## , wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; X is a methylene or an oxygen atom; and the dotted bonds can be hydrogenated, or an acid addition salt of a compound thereof which is basic.
Claim 4
Dependent Claim
97 words
A compound of the formula ##STR19## , wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; X is a methylene or an oxygen atom; and the dotted bonds can be hydrogenated, or an acid addition salt of a compound thereof which is basic.
Claim 5
Dependent Claim
91 words
A compound of the formula ##STR20## , wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound fthereof which is basic.
Claim 6
Dependent Claim
91 words
A compound of the formula ##STR20## , wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound fthereof which is basic.
Claim 7
Dependent Claim
90 words
A compound of the formula ##STR21## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 8
Dependent Claim
90 words
A compound of the formula ##STR21## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 9
Dependent Claim
90 words
A compound of the formula ##STR22## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 10
Dependent Claim
90 words
A compound of the formula ##STR22## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 11
Dependent Claim
90 words
A compound of the formula ##STR23## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 12
Dependent Claim
90 words
A compound of the formula ##STR23## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 13
Dependent Claim
90 words
A compound of the formula ##STR24## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 14
Dependent Claim
90 words
A compound of the formula ##STR24## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 15
Dependent Claim
90 words
A compound of the formula ##STR25## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 16
Dependent Claim
90 words
A compound of the formula ##STR25## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; and X is a methylene or an oxygen atom; or an acid addition salt of a compound thereof which is basic.
Claim 17
Dependent Claim
52 words
A compound of the formula ##STR26## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 7 , R 8 and R 9 , independently, are hydrogen or methyl; and X is methylene or an oxygen atom, or an acid addition salt of a compound thereof which is basic.
Claim 18
Dependent Claim
52 words
A compound of the formula ##STR26## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 7 , R 8 and R 9 , independently, are hydrogen or methyl; and X is methylene or an oxygen atom, or an acid addition salt of a compound thereof which is basic.
Claim 19
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-piperidine.
Claim 20
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3-methyl-piperidine.
Claim 21
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-morpholine.
Claim 22
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2,6-dimethyl-morpholine.
Claim 23
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-decahydroquinoline.
Claim 24
Dependent Claim
8 words
A compound in accordance with claim 1, 2-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-1,2,3,4-tetrahydroisoquinoline
Claim 25
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3,5-dimethyl-piperidine-1-oxide.
Claim 26
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2,4-dimethyl-piperidine-1-oxide.
Claim 27
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2,5-dimethyl-piperidine-1-oxide.
Claim 28
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3,5-dimethyl-piperidine-1-oxide.
Claim 29
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3,4-dimethyl-piperidine-1-oxide.
Claim 30
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3-ethyl-piperidine-1-oxide.
Claim 31
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3-ethyl-4-methyl-piperidine-1-oxide.
Claim 32
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2,4,6-trimethyl-piperidine-1-oxide.
Claim 33
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3,3-dimethyl-piperidine-1-oxide.
Claim 34
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-2-ethyl-piperidine.
Claim 35
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-3-methyl-piperidine.
Claim 36
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-3-ethyl-piperidine.
Claim 37
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-2,6-dimethyl-piperidine.
Claim 38
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-2,4-dimethyl-piperidine.
Claim 39
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-2,5-dimethyl-piperidine.
Claim 40
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-5-ethyl-2-methyl-piperidine.
Claim 41
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-3,5-dimethyl-piperidine.
Claim 42
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2-methyl-piperidine.
Claim 43
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-4-methyl-piperidine.
Claim 44
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-4-ethyl-piperidine.
Claim 45
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2,6-dimethyl-piperidine.
Claim 46
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-1,2,3,4-tetrahydroquinoline.
Claim 47
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-4-ethyl-piperidine.
Claim 48
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-3,4-dimethyl-piperidine.
Claim 49
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-3-ethyl-4-methyl-piperidine.
Claim 50
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-2,4,6-trimethyl-piperidine.
Claim 51
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-3,3-dimethyl-piperidine.
Claim 52
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-2,6-dimethyl-morpholine-4-oxide.
Claim 53
Dependent Claim
8 words
A compound in accordance with claim 1, 2-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-decahydroquinoline.
Claim 54
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(p-Tert.butyl-phenyl)-2,3-dimethyl-2-propenyl]-2,6-dimethyl-morpholine.
Claim 55
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2-ethyl-piperidine.
Claim 56
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3-ethyl-piperidine.
Claim 57
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2,4-dimethyl-piperidine.
Claim 58
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2,5-dimethyl-piperidine.
Claim 59
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-5-ethyl-2-methyl-piperidine.
Claim 60
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3,5-dimethyl-piperidine.
Claim 61
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3,4-dimethyl-piperidine.
Claim 62
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3-ethyl-4-methyl-piperidine.
Claim 63
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2,4,6-trimethyl-piperidine.
Claim 64
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3,3-dimethyl-piperidine.
Claim 65
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2,3-dimethyl-propyl]-piperidine.
Claim 66
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-1,2-dimethyl-propyl]-piperidine.
Claim 67
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-piperidine.
Claim 68
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-2,6-dimethyl-morpholine.
Claim 69
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2,3-dimethyl-2-propenyl]-piperidine.
Claim 70
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-2-propenyl]-piperidine.
Claim 71
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-2-propenyl]-3-methyl-piperidine.
Claim 72
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-2-propenyl]-2,6-dimethyl-morpholine.
Claim 73
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-phenyl)-2-methyl-propyl]-3,3-dimethyl-piperidine-1-oxide.
Claim 74
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-2,6-dimethyl-morpholine.
Claim 75
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-piperidine.
Claim 76
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-3-methyl-piperidine.
Claim 77
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-2,6-dimethyl-morpholine-4-oxide.
Claim 78
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-piperidine-1-oxide.
Claim 79
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-3-methyl-piperidine-1-oxide.
Claim 80
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(p-Tert.butyl-phenyl)-2-methyl-propyl]-morpholine-4-oxide.
Claim 81
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-1,2,3-trimethyl-2-propenyl]-piperidine.
Claim 82
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-1,2,3-trimethyl-propyl]-piperidine.
Claim 83
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-1,2-dimethyl-2-propenyl]-piperidine.
Claim 84
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-3-ethyl-piperidine.
Claim 85
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-3,5-dimethyl-piperidine.
Claim 86
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-3,4-dimethyl-piperidine.
Claim 87
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-3-ethyl-4-methyl-piperidine.
Claim 88
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-3-ethyl-piperidine-1-oxide.
Claim 89
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-3,4-dimethyl-piperidine-1-oxide.
Claim 90
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-3,5-dimethyl-piperidine-1-oxide.
Claim 91
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-2,6-dimethyl-morpholine-4-oxide.
Claim 92
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-piperidine-1-oxide.
Claim 93
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2-methyl-2-propenyl]-piperidine-1-oxide.
Claim 94
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-2-propenyl]-3-methyl-piperidine-1-oxide.
Claim 95
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2,3-dimethyl-2-propenyl]-3-methyl-piperidine.
Claim 96
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2,3-dimethyl-2-propenyl]-3,5-dimethyl-piperidine.
Claim 97
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2,3-dimethyl-propyl]-3-methyl-piperidine.
Claim 98
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(p-Tert.butyl-phenyl)-2,3-dimethyl-propyl]-3,5-dimethyl-piperidine.
Claim 99
Dependent Claim
8 words
A compound in accordance with claim 1, 4-[3-(p-Tert.butyl-phenyl)-2,3-dimethyl-propyl]-2,6-dimethyl-morpholine.
Claim 100
Dependent Claim
8 words
A compound in accordance with claim 1, 1-[3-(4-Tert.butyl-cyclohexyl)-2-methyl-propyl]-3-methyl-piperidine-1-oxide.
Claim 101
Dependent Claim
116 words
A fungicidal composition comprising an effective amount of at least one compound of the formula ##STR27## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; X is a methylene or an oxygen atom; z is zero or 1; and the dotted bonds can be hydrogenated, or an acid addition salt of a compound thereof which is basic and an inert carrier material.
Claim 102
Dependent Claim
116 words
A fungicidal composition comprising an effective amount of at least one compound of the formula ##STR27## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms, and two of R 4 , R 5 and R 6 can each be bonded to the same carbon atom or together can form a fused alicyclic or aromatic six-membered ring; X is a methylene or an oxygen atom; z is zero or 1; and the dotted bonds can be hydrogenated, or an acid addition salt of a compound thereof which is basic and an inert carrier material.
Claim 103
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-piperidine.
Claim 104
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3-methyl-piperidine.
Claim 105
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-morpholine.
Claim 106
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2,6-dimethyl-morpholine.
Claim 107
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-decahydroquinoline.
Claim 108
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 2-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-1,2,3,4-tetrahydroisoquinoline.
Claim 109
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3,5-dimethyl-piperidine-1-oxide.
Claim 110
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2,4-dimethyl-piperidine-1-oxide.
Claim 111
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2,5-dimethyl-piperidine-1-oxide.
Claim 112
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3,5-dimethyl-piperidine-1-oxide.
Claim 113
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3,4-dimethyl-piperidine-1-oxide.
Claim 114
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3-ethyl-piperidine-1-oxide.
Claim 115
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3-ethyl-4-methyl-piperidine-1-oxide.
Claim 116
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2,4,6-trimethyl-piperidine-1-oxide.
Claim 117
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3,3-dimethyl-piperidine-1-oxide.
Claim 118
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-2-ethyl-piperidine.
Claim 119
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-3-methyl-piperidine.
Claim 120
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-3-ethyl-piperidine.
Claim 121
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-2,6-dimethyl-piperidine.
Claim 122
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-2,4-dimethyl-piperidine.
Claim 123
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl-2,5-dimethyl-piperidine.
Claim 124
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-5-ethyl-2-methyl-piperidine.
Claim 125
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-3,5-dimethyl-piperidine.
Claim 126
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2-methyl-piperidine.
Claim 127
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-4-methyl-piperidine.
Claim 128
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-4-ethyl-piperidine.
Claim 129
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2,6-dimethyl-piperidine.
Claim 130
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-1,2,3,4-tetrahydroquinoline.
Claim 131
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-4-ethyl-piperidine.
Claim 132
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-3,4-dimethyl-piperidine.
Claim 133
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-3-ethyl-4-methyl-piperidine.
Claim 134
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-2,4,6-trimethyl-piperidine.
Claim 135
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-3,3-dimethyl-piperidine.
Claim 136
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-2,6-dimethyl-morpholine-4-oxide.
Claim 137
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 2-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-decahydroisoquinoline.
Claim 138
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(p-tert.butyl-phenyl)-2,3-dimethyl-2-propenyl]-2,6-dimethyl-morpholine.
Claim 139
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2-ethyl-piperidine.
Claim 140
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3-ethyl-piperidine.
Claim 141
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2,4-dimethyl-piperidine.
Claim 142
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2,5-dimethyl-piperidine.
Claim 143
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-5-ethyl-2-methyl-piperidine.
Claim 144
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3,5-dimethyl-piperidine.
Claim 145
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3,4-dimethyl-piperidine.
Claim 146
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3-ethyl-4-methyl-piperidine.
Claim 147
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2,4,6-trimethyl-piperidine.
Claim 148
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3,3-dimethyl-piperidine.
Claim 149
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.-butyl-phenyl)-2,2-dimethyl-propyl]-piperidine.
Claim 150
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.-butyl-phenyl)-1,2-dimethyl-propyl]-piperidine.
Claim 151
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-piperidine.
Claim 152
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-2,6-dimethyl-morpholine.
Claim 153
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2,3-dimethyl-2-propenyl]-piperidine.
Claim 154
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-2-propenyl]-piperidine.
Claim 155
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-2-propenyl]-3-methyl-piperidine.
Claim 156
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(4-tert.butyl-cyclohexyl)-2-methyl-2-propenyl]-2,6-dimethyl-morpholine.
Claim 157
Dependent Claim
11 words
A fungidical composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3,3-dimethyl-piperidine-1-oxide.
Claim 158
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-2,6-dimethyl-morpholine.
Claim 159
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-piperidine.
Claim 160
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-3-methyl-piperidine.
Claim 161
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-2,6-dimethyl-morpholine-4-oxide.
Claim 162
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-piperidine-1-oxide.
Claim 163
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-3-methyl-piperidine-1-oxide.
Claim 164
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(p-tert.butyl-phenyl)-2-methyl-propyl]-morpholine-4-oxide.
Claim 165
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-1,2,3-trimethyl-2-propenyl]-piperidine.
Claim 166
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-1,2,3-trimethyl-propyl]-piperidine.
Claim 167
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-1,2-dimethyl-2-propenyl]-piperidine.
Claim 168
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-3-ethyl-piperidine.
Claim 169
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-3,5-dimethyl-piperidine.
Claim 170
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-3,4-dimethyl-piperidine.
Claim 171
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-3-ethyl-4-methyl-piperidine.
Claim 172
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-3-ethyl-piperidine-1-oxide.
Claim 173
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-3,4-dimethyl-piperidine-1-oxide.
Claim 174
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-3,5-dimethyl-piperidine-1-oxide.
Claim 175
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-2,6-dimethyl-morpholine-4-oxide.
Claim 176
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-propyl]-piperidine-1-oxide.
Claim 177
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2-methyl-2-propenyl]-piperidine-1-oxide.
Claim 178
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(4-tert.butyl-cyclohexyl)-2-methyl-2-propenyl]-3-methyl-piperidine-1-oxide.
Claim 179
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2,3-dimethyl-2-propenyl]-3-methyl-piperidine.
Claim 180
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2,3-dimethyl-2-propenyl]-3,5-dimethyl-piperidine.
Claim 181
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2,3-dimethyl-propyl]-3-methyl-piperidine.
Claim 182
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 1-[3-(p-tert.butyl-phenyl)-2,3-dimethyl-propyl]-3,5-dimethyl-piperidine.
Claim 183
Dependent Claim
11 words
A fungicidal composition, in accordance with claim 92, which contains 4-[3-(p-tert.butyl-phenyl)-2,3-dimethyl-propyl]-2,6-dimethyl-morpholine.
Claim 184
Dependent Claim
44 words
A compound of the formula ##STR28## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms; and the acid addition salts thereof.
Claim 185
Dependent Claim
44 words
A compound of the formula ##STR28## wherein R 1 and R 3 , independently, are hydrogen or methyl; R 4 , R 5 and R 6 , independently, are hydrogen or alkyl of 1 to 4 carbon atoms; and the acid addition salts thereof.
References Cited (Backward Citations)
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1983-12-23 | 1984-06-23 | 1984-12-23 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1987-12-23 | 1988-06-23 | 1988-12-23 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1991-12-23 | 1992-06-23 | 1992-12-23 | $7700.00 | Window Closed / Lapsed |