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US4238501A Expired / Lapsed US ⏱️ 0.0 years remaining

Combating arthropods with 2- and 4-substituted-chromanes

Assignee: Bayer AG
•
Filing: 1979-08-15
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Granted: 1980-12-09
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Expires: 1999-08-15
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Abstract

Abstract Chromane derivatives of the formula <IMAGE> in which R1 to R4, which need not be identical, each represents hydrogen, an optionally substituted alkyl, alkenyl, cycloalkyl, aryl, aralkyl or alkoxycarbonyl radical, carboxyl or aminoalkyl, R2 can alternatively represent amino or optionally substituted dialkylamino, or R1 and R2 conjointly with the adjoining carbon atoms can form an optionally substituted carbocyclic or heterocyclic ring, R5 to R8, which need not be identical, each represents hydrogen, halogen, hydroxyl, nitro, cyano, carboxyl, an optionally substituted alkyl, alkenyl, cycloalkyl, aryl, aralkyl, alkoxy, aralkoxy, aryloxy, alkoxycarbonyl, alkylamino or dialkylamino radical, amino or acylamino, and two of the radicals, which are in the o-position to one another, can represent tetramethylene or the radical -CH=CH-CH=CH-, and X represents OH or the -NR9R10 radical, wherein R9 and R10, which may be identical or different, each represents hydrogen or optionally substituted alkyl, alkenyl, cycloalkyl, aryl or aralkyl, or R9 and R10 conjointly with the adjoining nitrogen atom form a ring which optionally contains one or more further hetero-atoms, or optionally, when X is -NR9R10, a salt thereof, in which X is a hydroxy or amino radical, and R1 to R8 can be hydrogen or various organic radicals, or salts thereof possess arthropodicidal properties. Those compounds wherein R1 and R2 conjointly with the adjoining carbon atoms forms a carbocyclic or heterocyclic ring are new.

Inventors

  • 👤 Hans-Joachim Kabbe
  • 👤 Arno Widdig
  • 👤 Wilhelm Stendel
  • 👤 Peter Roessler

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-03 13:51
CPC Classifications
C; C07; C07D; C07D491/00; C07D491/02; C07D491/10; A; A01; A01N; A01N43/00; A01N43/02; A01N43/04; A01N43/14; A01N43/16; A01N43/34; A01N43/36; A01N43/40; A01N43/90; C07D311/00; C07D311/02; C07D311/04; C07D311/22; C07D311/24; C07D311/96

Claims Analysis

Total Claims: 5
Claim 1
Independent Claim 124 words
A compound of the formula ##STR11## in which R 3 and R 4 , which need not be identical, each represents hydrogen, an optionally substituted alkyl, alkenyl, cycloalkyl, aryl, aralkyl or alkoxycarbonyl radical, carboxyl or aminoalkyl, R 1 and R 2 conjointly with the adjoining carbon atoms can form an optionally substituted carbocyclic, R 5 to R 8 , which need not be identical, each represents hydrogen, halogen, hydroxyl, nitro, cyano, carboxyl, an optionally substituted alkyl, alkenyl, cycloalkyl, aryl, aralkyl, alkoxy, aralkoxy, aryloxy, alkoxycarbonyl, alkylamino or dialkylamino radical, amino or acylamino, X represents the --NR 9 R 10 radical, wherein R 9 and R 10 , which may be identical or different, each represents hydrogen or optionally substituted alkyl, alkenyl, cycloalkyl, aryl or aralkyl.
Claim 2
Dependent Claim 124 words
A compound of the formula ##STR11## in which R 3 and R 4 , which need not be identical, each represents hydrogen, an optionally substituted alkyl, alkenyl, cycloalkyl, aryl, aralkyl or alkoxycarbonyl radical, carboxyl or aminoalkyl, R 1 and R 2 conjointly with the adjoining carbon atoms can form an optionally substituted carbocyclic, R 5 to R 8 , which need not be identical, each represents hydrogen, halogen, hydroxyl, nitro, cyano, carboxyl, an optionally substituted alkyl, alkenyl, cycloalkyl, aryl, aralkyl, alkoxy, aralkoxy, aryloxy, alkoxycarbonyl, alkylamino or dialkylamino radical, amino or acylamino, X represents the --NR 9 R 10 radical, wherein R 9 and R 10 , which may be identical or different, each represents hydrogen or optionally substituted alkyl, alkenyl, cycloalkyl, aryl or aralkyl.
Claim 3
Dependent Claim 16 words
A compound according to claim 1, wherein the chromane derivative is 4-dimethylamino-2,2-pentamethylene-chromane of the formula ##STR12##
Claim 4
Dependent Claim 28 words
A method of combating arthropods which comprises applying to the arthropods, or to a habitat thereof, an arthropodicidally effective amount of a chromane derivative according to claim 1.
Claim 5
Dependent Claim 18 words
An arthropodicidal composition comprising a diluent plus an arthropodicidally effective amount of a compound according to claim 1.

References Cited (Backward Citations)

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USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1983-12-09 1984-06-09 1984-12-09 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1987-12-09 1988-06-09 1988-12-09 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1991-12-09 1992-06-09 1992-12-09 $7700.00 Window Closed / Lapsed

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