US4182330A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Means for administering amphipathic medicament
Assignee: Alza Corp
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Filing: 1977-07-25
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Granted: 1980-01-08
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Expires: 1997-07-25
Abstract
Abstract Means for administering an amphipathic medicament by micelle solubilization is disclosed. The micelle consists of a nonionic surfactant medicament adduct. The adduct is coated onto an osmotically effective solute and housed in an osmotic therapeutic system for administering the medicament in a therapeutically effective amount over a prolonged period of time.
Inventors
- 👤 Alan S. Michaels
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-10-23 15:17
CPC Classifications
A; A61; A61K; A61K9/00; A61K9/10; A61K9/107; A61K9/1075; A61K9/0002; A61K9/0004
Claims Analysis
Total Claims: 11
Claim 1
Independent Claim
196 words
An osmotic therapeutic system for the controlled dispensing of drug to a biological environment of use, said system comprising: (a) a shaped wall formed of a non-toxic semipermeable material that maintains its integrity during the drug dispensing period and which material is permeable to the passage of an external fluid in the environment and substantially impermeable to the passage of drug, the wall surrounding and forming; (b) a compartment; (c) a micelle comprising an amphipathic drug pharmaceutically acceptable surfactant adduct which adduct is coated onto an osmotically effective solute that exhibits an osmotic pressure gradient across the wall against the fluid housed in the compartment; (d) a passageway in the wall communicating with the compartment and the exterior of the system, and; (e) wherein in operation when the system is in the environment, fluid from the environment is imbibed through the wall into the compartment in a tendency towards osmotic equilibrium at a rate determined by the permeability of the wall and the osmotic pressure gradient across the wall, thereby continuously forming a solution of adduct, which solution containing the drug is dispensed through the passageway at a controlled rate over a prolonged period of time.
Claim 2
Dependent Claim
196 words
An osmotic therapeutic system for the controlled dispensing of drug to a biological environment of use, said system comprising: (a) a shaped wall formed of a non-toxic semipermeable material that maintains its integrity during the drug dispensing period and which material is permeable to the passage of an external fluid in the environment and substantially impermeable to the passage of drug, the wall surrounding and forming; (b) a compartment; (c) a micelle comprising an amphipathic drug pharmaceutically acceptable surfactant adduct which adduct is coated onto an osmotically effective solute that exhibits an osmotic pressure gradient across the wall against the fluid housed in the compartment; (d) a passageway in the wall communicating with the compartment and the exterior of the system, and; (e) wherein in operation when the system is in the environment, fluid from the environment is imbibed through the wall into the compartment in a tendency towards osmotic equilibrium at a rate determined by the permeability of the wall and the osmotic pressure gradient across the wall, thereby continuously forming a solution of adduct, which solution containing the drug is dispensed through the passageway at a controlled rate over a prolonged period of time.
Claim 3
Dependent Claim
32 words
The osmotic therapeutic system for the controlled dispensing of beneficial drug according to claim 1 wherein the drug is a member selected from the group consisting of locally and systemically acting drugs.
Claim 4
Dependent Claim
32 words
The osmotic therapeutic system for the controlled dispensing of beneficial drug according to claim 1, wherein the micelle is a micellar aggregate consisting essentially of an amphipathic drug and a nonionic surfactant.
Claim 5
Dependent Claim
45 words
The osmotic therapeutic system for the controlled dispensing of beneficial drug according to claim 1, wherein the amphipathic drug is a member selected from the group consisting of central nervous system, hypnotic, sedative, tranquilizer, anticonvulsant, antiparkinson, analgesic, anesthetic, antispasmodic, antiviral, antiulcer, hormonal and antimicrobial drugs.
Claim 6
Dependent Claim
34 words
The osmotic therapeutic system for the controlled dispensing of beneficial drug according to claim 1 wherein the micelle consists of 10 parts to 300 parts by weight of surfactant per 100 parts of drug.
Claim 7
Dependent Claim
23 words
The osmotic therapeutic system for the controlled dispensing of beneficial drug according to claim 1 wherein the drug is a pharmaceutically acceptable steroid.
Claim 8
Dependent Claim
166 words
A medicament for the management of cardiac decompensation, said medicament consisting essentially of (a) an adduct consisting of a digitaloid drug and a pharmaceutically acceptable nonionic surfactant, and (b) an osmotically effective solute which exhibits an osmotic pressure gradient across a semipermeable wall against an external fluid coated with the adduct, said medicament housed in an osmotic delivery system which system comprises (1) a shaped semipermeable wall permeable to the passage of fluid and impermeable to the passage of medicament, (2) the wall surrounding and forming a compartment housing the medicament, (3) a passageway in the wall communicating with the compartment and the exterior of the system, and (4) wherein in operation when the system is in a biological environment fluid from the environment is imbibed through the wall into the compartment forming a solution of adduct which solution containing the drug is released through the passageway at a controlled rate over a prolonged period of time thereby administering the drug for its intended beneficial effect.
Claim 9
Dependent Claim
166 words
A medicament for the management of cardiac decompensation, said medicament consisting essentially of (a) an adduct consisting of a digitaloid drug and a pharmaceutically acceptable nonionic surfactant, and (b) an osmotically effective solute which exhibits an osmotic pressure gradient across a semipermeable wall against an external fluid coated with the adduct, said medicament housed in an osmotic delivery system which system comprises (1) a shaped semipermeable wall permeable to the passage of fluid and impermeable to the passage of medicament, (2) the wall surrounding and forming a compartment housing the medicament, (3) a passageway in the wall communicating with the compartment and the exterior of the system, and (4) wherein in operation when the system is in a biological environment fluid from the environment is imbibed through the wall into the compartment forming a solution of adduct which solution containing the drug is released through the passageway at a controlled rate over a prolonged period of time thereby administering the drug for its intended beneficial effect.
Claim 10
Dependent Claim
20 words
The medicament for the management of cardiac decompensation according to claim 7 wherein the digitaloid drug is a cardiac glycoside.
Claim 11
Dependent Claim
36 words
The medicament for the management of cardiac decompensation according to claim 7 wherein the digitaloid drug is a member selected from the group consisting of acetyldigitoxin, deslanoside, digitalis, digitoxin, digoxin, gitalin, lanatoside, ovabain and mixtures thereof.
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USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1983-01-07 | 1983-07-09 | 1984-01-08 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1987-01-07 | 1987-07-09 | 1988-01-08 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1991-01-07 | 1991-07-09 | 1992-01-08 | $7700.00 | Window Closed / Lapsed |