US4169205A
Expired / Lapsed
US
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Imidazole derivatives of 6,11-dihydrodibenz[b,e]oxepines and 6,11-dihydrodibenz[b,e]thiepines
Assignee: ER Squibb and Sons LLC
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Filing: 1978-10-25
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Granted: 1979-09-25
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Expires: 1998-10-25
Abstract
Abstract New imidazole derivatives of 6,11-dihydrodibenz[b,e]oxepines and 6,11-dihydrodibenz[b,e]thiepines have the general formula ##STR1## They and the salts thereof are useful as antifungal and antibacterial agents.
Inventors
- 👤 Hans Hoehn
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-04 14:16
CPC Classifications
C; C07; C07D; C07D231/00; C07D231/02; C07D231/10; C07D231/12; C07D233/00; C07D233/54; C07D233/56; C07D249/00; C07D249/02; C07D249/08
Claims Analysis
Total Claims: 14
Claim 1
Independent Claim
72 words
A compound of the formula ##STR18## wherein X is oxygen or sulfur; R 1 and R 2 each is hydrogen, halogen, hydroxy, trifluoromethyl, lower alkyl, lower alkoxy, lower alkylthio, nitro or the group ##STR19## R 3 and R 4 each is hydrogen, lower alkyl, phenyl or substituted phenyl wherein the phenyl bears one halogen, hydroxy, lower alkoxy, lower alkyl, lower alkylthio, cyano or nitro; and non-toxic, physiologically acceptable acid addition salts thereof.
Claim 2
Dependent Claim
72 words
A compound of the formula ##STR18## wherein X is oxygen or sulfur; R 1 and R 2 each is hydrogen, halogen, hydroxy, trifluoromethyl, lower alkyl, lower alkoxy, lower alkylthio, nitro or the group ##STR19## R 3 and R 4 each is hydrogen, lower alkyl, phenyl or substituted phenyl wherein the phenyl bears one halogen, hydroxy, lower alkoxy, lower alkyl, lower alkylthio, cyano or nitro; and non-toxic, physiologically acceptable acid addition salts thereof.
Claim 3
Dependent Claim
18 words
A compound as in claim 1 wherein R 1 is hydrogen or halogen and R 2 is hydrogen.
Claim 4
Dependent Claim
17 words
A compound as in claim 1 wherein R 1 and R 2 each is hydrogen or halogen.
Claim 5
Dependent Claim
15 words
A compound as in claim 1 wherein R 1 and R 2 each is hydrogen.
Claim 6
Dependent Claim
16 words
A compound as in claim 1 wherein R 1 is halogen and R 2 is hydrogen.
Claim 7
Dependent Claim
11 words
A compound as in claim 5 wherein the halogen is chlorine.
Claim 8
Dependent Claim
24 words
A compound as in claim 1 wherein R 1 is ##STR20## and R 3 and R 4 each is hydrogen, lower alkyl or phenyl.
Claim 9
Dependent Claim
10 words
A compound as in claim 1 wherein X is oxygen.
Claim 10
Dependent Claim
10 words
A compound as in claim 1 wherein X is sulfur.
Claim 11
Dependent Claim
19 words
A compound as in claim 1 wherein X is oxygen; R 1 is 2-chloro; and R 2 is hydrogen.
Claim 12
Dependent Claim
19 words
A compound as in claim 1 wherein X is oxygen and R 1 and R 2 each is hydrogen.
Claim 13
Dependent Claim
19 words
A compound as in claim 1 wherein X is sulfur and R 1 and R 2 each is hydrogen.
Claim 14
Dependent Claim
19 words
A compound as in claim 1 wherein X is sulfur; R 1 is 2-chloro; and R 2 is hydrogen.
References Cited (Backward Citations)
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Cited
US3647816A
Cited
GB1299246A
Cited
US3764609A
Cited
US3778447A
Cited
US4049418A
Cited
US4021561A
Cited
US4112112A
Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1982-09-24 | 1983-03-26 | 1983-09-25 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1986-09-24 | 1987-03-26 | 1987-09-25 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1990-09-24 | 1991-03-26 | 1991-09-25 | $7700.00 | Window Closed / Lapsed |