US4143155A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Sulfonylglycolic anilide fungicides
Assignee: Novartis Corp
•
Filing: 1977-09-12
•
Granted: 1979-03-06
•
Expires: 1997-09-12
Abstract
Abstract Compounds of the formula I ##STR1## wherein R 1 represents C 1 -C 4 alkyl, C 1 -C 4 alkoxy or halogen, R 2 represents hydrogen, C 1 -C 3 alkyl, C 1 -C 4 alkoxy or halogen, R 3 represents hydrogen, C 1 -C 3 alkyl or halogen, and R 4 represents hydrogen or methyl, with the proviso that the total number of carbon atoms contained by the substituents R 1 , R 2 , R 3 and R 4 does not exceed 8, X represents ##STR2## and R 5 represents hydrogen or methyl and R 6 represents C 1 -C 6 alkyl which is unsubstituted or substituted by halogen or represents C 2 -C 4 alkenyl or C 3 -C 6 cycloalkyl or the group --N(R 7 )R 8 , in which R 7 represents hydrogen or C 1 -C 4 alkyl and R 8 represents C 1 -C 6 alkyl which is unsubstituted or substituted by halogen, which are useful in combatting microorganisms in particular phytopathogenic fungi.
Inventors
- 👤 Adolf Hubele
- 👤 Wolfgang Eckhardt
- 👤 Walter Kunz
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-05 11:45
CPC Classifications
C; C07; C07D; C07D307/00; C07D307/02; C07D307/26; C07D307/30; C07D307/32; C07D307/33; A; A01; A01N; A01N41/00; A01N41/02; A01N41/04; A01N41/08; A01N43/00; A01N43/02; A01N43/04; A01N43/06; A01N43/08
Claims Analysis
Total Claims: 25
Claim 1
Independent Claim
160 words
A compound of the formula I ##STR22## wherein R 1 represents C 1 -C 4 alkyl, C 1 -C 4 alkoxy or halogen, R 2 represents hydrogen, C 1 -C 3 alkyl, C 1 -C 4 alkoxy or halogen, R 3 represents hydrogen, C 1 -C 3 alkyl or halogen, and R 4 represents hydrogen or methyl, with the proviso that the total number of carbon atoms contained by the substituents R 1 , R 2 , R 3 and R 4 does not exceed 8, X represents ##STR23## R 5 represents hydrogen or methyl and R 6 represents C 1 -C 6 alkyl which is unsubstituted or substituted by halogen or represents C 2 -C 4 alkenyl or C 3 -C 6 cycloalkyl or the group --N(R 7 )R 8 , in which R 7 represents hydrogen or C 1 -C 4 alkyl and R 8 represents C 1 -C 6 alkyl which is unsubstituted or substituted by halogen.
Claim 2
Dependent Claim
160 words
A compound of the formula I ##STR22## wherein R 1 represents C 1 -C 4 alkyl, C 1 -C 4 alkoxy or halogen, R 2 represents hydrogen, C 1 -C 3 alkyl, C 1 -C 4 alkoxy or halogen, R 3 represents hydrogen, C 1 -C 3 alkyl or halogen, and R 4 represents hydrogen or methyl, with the proviso that the total number of carbon atoms contained by the substituents R 1 , R 2 , R 3 and R 4 does not exceed 8, X represents ##STR23## R 5 represents hydrogen or methyl and R 6 represents C 1 -C 6 alkyl which is unsubstituted or substituted by halogen or represents C 2 -C 4 alkenyl or C 3 -C 6 cycloalkyl or the group --N(R 7 )R 8 , in which R 7 represents hydrogen or C 1 -C 4 alkyl and R 8 represents C 1 -C 6 alkyl which is unsubstituted or substituted by halogen.
Claim 3
Dependent Claim
35 words
A compound according to claim 1 wherein R 1 represents methyl, R 2 represents methyl or chlorine in the 6-position, R 3 represents hydrogen, chlorine, bromine or methyl and R 4 represents hydrogen or methyl.
Claim 4
Dependent Claim
21 words
A compound according to claim 1 wherein R 6 represents C 1 -C 4 alkyl or the group NHR 8 .
Claim 5
Dependent Claim
11 words
A compound according to claim 1 wherein R 5 represents hydrogen.
Claim 6
Dependent Claim
89 words
A compound according to claim 1 wherein R 1 represents metyl or methoxy, R 2 represents methyl, ethyl or chlorine, R 3 represents hydrogen, methyl, chlorine or bromine, R 4 represents hydrogen or methyl, R 5 represents hydrogen and R 6 represents C 1 -C 6 -alkyl which is unsubstituted or substituted by halogen, or represents vinyl, allyl, cyclohexyl or the group N(R 7 )R 8 in which R 7 represents hydrogen, methyl or ethyl and R 8 represents methyl or ethyl which is unsubstituted or substituted by chlorine.
Claim 7
Dependent Claim
27 words
A compound according to claim 2 wherein R 5 represents hydrogen and R 6 l represents C 1 -C 4 alkyl or the group NHR 8 .
Claim 8
Dependent Claim
9 words
A compound according to claim 1 which is N-(1'-methoxycarbonylethyl)-N-(methylsulphonoxy-acetyl)-2,6-dimethylaniline.
Claim 9
Dependent Claim
18 words
A compound according to claim 1 selected from the group consisting of N-(1'-methoxycarbonylethyl)-N-(ethylsulphonoxy-acetyl)-2,6-dimethylaniline, N-(1'-methoxycarbonylethyl)-N-(n-propylsulphonoxy-acetyl)-2,6-dimethylaniline, N-(1'-methoxycarbonylethyl)-N-(n-butylsulphonoxy-acetyl)-2,6-dimethylaniline, N-(1'-methoxycarbonylethyl)-N-(methylaminosulphonoxy-acetyl)-2,6-dimethylaniline, and N-(1'-methoxycarbonylethyl)-N-(methylsulphonoxy-acetyl)-2,3,6-trimethylaniline.
Claim 10
Dependent Claim
37 words
A phytopathogenic fungicidal composition containing as active ingredient a phytopathogenic fungicidally effective amount of a compound according to claim 1 together with a solid extender and optionally a surfactant or with a liquid diluent and a surfactant.
Claim 11
Dependent Claim
37 words
A phytopathogenic fungicidal composition containing as active ingredient a phytopathogenic fungicidally effective amount of a compound according to claim 2 together with a solid extender and optionally a surfactant or with a liquid diluent and a surfactant.
Claim 12
Dependent Claim
37 words
A phytopathogenic fungicidal composition containing as active ingredient a phytopathogenic fungicidally effective amount of a compound according to claim 3 together with a solid extender and optionally a surfactant or with a liquid diluent and a surfactant.
Claim 13
Dependent Claim
37 words
A phytopathogenic fungicidal composition containing as active ingredient a phytopathogenic fungicidally effective amount of a compound according to claim 4 together with a solid extender and optionally a surfactant or with a liquid diluent and a surfactant.
Claim 14
Dependent Claim
37 words
A phytopathogenic fungicidal composition containing as active ingredient a phytopathogenic fungicidally effective amount of a compound according to claim 5 together with a solid extender and optionally a surfactant or with a liquid diluent and a surfactant.
Claim 15
Dependent Claim
37 words
A phytopathogenic fungicidal composition containing as active ingredient a phytopathogenic fungicidally effective amount of a compound according to claim 6 together with a solid extender and optionally a surfactant or with a liquid diluent and a surfactant.
Claim 16
Dependent Claim
37 words
A phytopathogenic fungicidal composition containing as active ingredient a phytopathogenic fungicidally effective amount of a compound according to claim 7 together with a solid extender and optionally a surfactant or with a liquid diluent and a surfactant.
Claim 17
Dependent Claim
37 words
A phytopathogenic fungicidal composition containing as active ingredient a phytopathogenic fungicidally effective amount of a compound according to claim 8 together with a solid extender and optionally a surfactant or with a liquid diluent and a surfactant.
Claim 18
Dependent Claim
25 words
A method of combatting phytopathogenic fungi which comprises applying thereto or to the locus thereof an effective amount of a compound according to claim 1.
Claim 19
Dependent Claim
25 words
A method of combatting phytopathogenic fungi which comprises applying thereto or to the locus thereof an effective amount of a compound according to claim 2.
Claim 20
Dependent Claim
25 words
A method of combatting phytopathogenic fungi which comprises applying thereto or to the locus thereof an effective amount of a compound according to claim 3.
Claim 21
Dependent Claim
25 words
A method of combatting phytopathogenic fungi which comprises applying thereto or to the locus thereof an effective amount of a compound according to claim 4.
Claim 22
Dependent Claim
25 words
A method of combatting phytopathogenic fungi which comprises applying thereto or to the locus thereof an effective amount of a compound according to claim 5.
Claim 23
Dependent Claim
25 words
A method of combatting phytopathogenic fungi which comprises applying thereto or to the locus thereof an effective amount of a compound according to claim 6.
Claim 24
Dependent Claim
25 words
A method of combatting phytopathogenic fungi which comprises applying thereto or to the locus thereof an effective amount of a compound according to claim 7.
Claim 25
Dependent Claim
25 words
A method of combatting phytopathogenic fungi which comprises applying thereto or to the locus thereof an effective amount of a compound according to claim 8.
References Cited (Backward Citations)
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1982-03-05 | 1982-09-04 | 1983-03-06 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1986-03-05 | 1986-09-04 | 1987-03-06 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1990-03-05 | 1990-09-04 | 1991-03-06 | $7700.00 | Window Closed / Lapsed |