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US4137404A Expired / Lapsed US ⏱️ 0.0 years remaining

Synthesis of tryptophans

Assignee: Hoffmann La Roche Inc
•
Filing: 1977-12-20
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Granted: 1979-01-30
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Expires: 1997-12-20
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Abstract

Abstract A process is disclosed for preparing racemic and optically pure tryptophans through novel intermediates.

Inventors

  • 👤 Andrew D. Batcho
  • 👤 Willy Leimgruber

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-10-26 15:29
CPC Classifications
C; C07; C07D; C07D309/00; C07D309/34; C07D309/36; C07D309/38; C07D209/00; C07D209/02; C07D209/04; C07D209/10; C07D209/18; C07D209/20; C07D263/00; C07D263/02; C07D263/30; C07D263/34; C07D263/36; C07D263/42

Claims Analysis

Total Claims: 4
Claim 1
Independent Claim 36 words
A compound of the formula: ##STR4## wherein R 1 and R 16 individually are halogen, lower alkyl, hydroxy, lower alkoxy, aralkyloxy, amino, trihalomethyl or hydrogen and R 9 is lower alkyl, aryl, hydrogen or halo-lower alkyl.
Claim 2
Dependent Claim 36 words
A compound of the formula: ##STR4## wherein R 1 and R 16 individually are halogen, lower alkyl, hydroxy, lower alkoxy, aralkyloxy, amino, trihalomethyl or hydrogen and R 9 is lower alkyl, aryl, hydrogen or halo-lower alkyl.
Claim 3
Dependent Claim 10 words
The compound of claim 1 wherein said compound is 4-[3-dimethylamino-2-(4-methyl-2-nitrophenyl)-2-propen-1-ylidene]-2-methyl-2-oxazolin-5-one.
Claim 4
Dependent Claim 10 words
The compound of claim 1 wherein said compound is 4-[3-dimethylamino-2-(2-nitrophenyl)-2-propen-1-ylidene]-2-methyl-2-oxazolin-5-one.

References Cited (Backward Citations)

US3949000A Cited
US3956304A Cited
US4073795A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1982-01-29 1982-07-31 1983-01-30 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1986-01-29 1986-07-31 1987-01-30 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1990-01-29 1990-07-31 1991-01-30 $7700.00 Window Closed / Lapsed

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