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US3980781A Expired / Lapsed US ⏱️ 0.0 years remaining

Fungicidal composition and method containing 2-amino-pyrimidines

Assignee: Imperial Chemical Industries Ltd
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Filing: 1971-12-13
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Granted: 1976-09-14
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Expires: 1991-12-13
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Abstract

Abstract Fungicidal pyrimidine derivatives and the use thereof in combatting plant diseases. Representative derivatives are 2-dimethylamino-4-methyl-5-n-pentyl-6-hydroxypyrimidine and 2-dimethylamino-4-methyl-5-n-propyl-6-hydroxypyrimidine.

Inventors

  • 👤 Brian Kenneth Snell
  • 👤 Richard Stewart Elias
  • 👤 Peter Frank Hilary Freeman

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-01 00:23
CPC Classifications
C; C07; C07D; C07D401/00; C07D401/02; C07D401/04; C07D239/00; C07D239/02; C07D239/24; C07D239/28; C07D239/46; C07D239/47; C07D401/12; C07D413/00; C07D413/02; C07D413/04; C07F; C07F3/00; C07F3/10; C07F3/103

Claims Analysis

Total Claims: 13
Claim 1
Independent Claim 92 words
A process for combatting powdery mildew which comprises applying to the locus of the plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine derivative of the formula: ##SPC26## or a salt thereof, wherein R 1 and R 2 are hydrogen or lower alkyl; R 3 is lower alkyl; R 4 is lower alkyl or lower alkenyl; X is oxygen or sulfur and R 5 is hydrogen.
Claim 2
Dependent Claim 92 words
A process for combatting powdery mildew which comprises applying to the locus of the plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine derivative of the formula: ##SPC26## or a salt thereof, wherein R 1 and R 2 are hydrogen or lower alkyl; R 3 is lower alkyl; R 4 is lower alkyl or lower alkenyl; X is oxygen or sulfur and R 5 is hydrogen.
Claim 3
Dependent Claim 94 words
A process for combatting powdery mildew which comprises applying to the locus of the plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine derivative of the formula: ##SPC27## or a salt thereof, wherein R 1 and R 2 are hydrogen, lower alkyl, or lower alkenyl; R 3 is lower alkyl; R 4 is lower alkyl or lower alkenyl; X is oxygen or sulfur and R 5 is hydrogen.
Claim 4
Dependent Claim 94 words
A process for combatting powdery mildew which comprises applying to the locus of the plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine derivative of the formula: ##SPC27## or a salt thereof, wherein R 1 and R 2 are hydrogen, lower alkyl, or lower alkenyl; R 3 is lower alkyl; R 4 is lower alkyl or lower alkenyl; X is oxygen or sulfur and R 5 is hydrogen.
Claim 5
Dependent Claim 44 words
A process according to claim 2 wherein R 1 is hydrogen, allyl, ethyl, propyl or butyl; R 2 is allyl, methyl, ethyl, propyl or butyl; R 3 is methyl or ethyl; R 4 is methyl, ethyl, propyl, butyl, or amyl; and X is oxygen.
Claim 6
Dependent Claim 67 words
A process for combatting powdery mildew which comprises applying to the locus of plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine compound, or salt thereof, selected from: 2-dimethylamino-4-methyl-5-n-pentyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-n-propyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-isopropylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-amino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-n-propylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-dimethylamino-4-ethyl-5-n-butyl-6-hydroxypyrimidine; 2-diethylamino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-diethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-ethyl-6-mercaptopyrimidine; 2-dimethylamino-4-methyl-5-n-butyl-6(2-dimethylaminoethylthio)pyrimidine; and 2-dimethylamino-4-methyl-5-n-butyl-6-(2-diethylaminoethylthio)pyrimidine.
Claim 7
Dependent Claim 67 words
A process for combatting powdery mildew which comprises applying to the locus of plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine compound, or salt thereof, selected from: 2-dimethylamino-4-methyl-5-n-pentyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-n-propyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-isopropylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-amino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-n-propylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-dimethylamino-4-ethyl-5-n-butyl-6-hydroxypyrimidine; 2-diethylamino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-diethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-ethyl-6-mercaptopyrimidine; 2-dimethylamino-4-methyl-5-n-butyl-6(2-dimethylaminoethylthio)pyrimidine; and 2-dimethylamino-4-methyl-5-n-butyl-6-(2-diethylaminoethylthio)pyrimidine.
Claim 8
Dependent Claim 12 words
A process according to claim 1 wherein the pyrimidine derivative is 2-dimethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine.
Claim 9
Dependent Claim 12 words
A process according to claim 1 wherein the pyrimidine derivative is 2-ethylamino-4-methyl-5-n-butyl-6-hyroxypyrimidine.
Claim 10
Dependent Claim 12 words
A process according to claim 1 wherein the plants are cucurbit plants.
Claim 11
Dependent Claim 15 words
A process according to claim 1 wherein the plants are cereal crops barley or wheat.
Claim 12
Dependent Claim 26 words
A fungicidal composition for combatting powdery mildew comprising, as a systemically active ingredient, a fungicidally effective amount of 2-ethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine and an inert carrier for said ingredient.
Claim 13
Dependent Claim 26 words
A fungicidal composition for combatting powdery mildew comprising, as a systemically active ingredient, a fungicidally effective amount of 2-ethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine and an inert carrier for said ingredient.

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1979-09-14 1980-03-15 1980-09-14 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1983-09-14 1984-03-15 1984-09-14 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1987-09-14 1988-03-15 1988-09-14 $7700.00 Window Closed / Lapsed

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