US3980781A
Expired / Lapsed
US
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Fungicidal composition and method containing 2-amino-pyrimidines
Assignee: Imperial Chemical Industries Ltd
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Filing: 1971-12-13
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Granted: 1976-09-14
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Expires: 1991-12-13
Abstract
Abstract Fungicidal pyrimidine derivatives and the use thereof in combatting plant diseases. Representative derivatives are 2-dimethylamino-4-methyl-5-n-pentyl-6-hydroxypyrimidine and 2-dimethylamino-4-methyl-5-n-propyl-6-hydroxypyrimidine.
Inventors
- 👤 Brian Kenneth Snell
- 👤 Richard Stewart Elias
- 👤 Peter Frank Hilary Freeman
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-01 00:23
CPC Classifications
C; C07; C07D; C07D401/00; C07D401/02; C07D401/04; C07D239/00; C07D239/02; C07D239/24; C07D239/28; C07D239/46; C07D239/47; C07D401/12; C07D413/00; C07D413/02; C07D413/04; C07F; C07F3/00; C07F3/10; C07F3/103
Claims Analysis
Total Claims: 13
Claim 1
Independent Claim
92 words
A process for combatting powdery mildew which comprises applying to the locus of the plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine derivative of the formula: ##SPC26## or a salt thereof, wherein R 1 and R 2 are hydrogen or lower alkyl; R 3 is lower alkyl; R 4 is lower alkyl or lower alkenyl; X is oxygen or sulfur and R 5 is hydrogen.
Claim 2
Dependent Claim
92 words
A process for combatting powdery mildew which comprises applying to the locus of the plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine derivative of the formula: ##SPC26## or a salt thereof, wherein R 1 and R 2 are hydrogen or lower alkyl; R 3 is lower alkyl; R 4 is lower alkyl or lower alkenyl; X is oxygen or sulfur and R 5 is hydrogen.
Claim 3
Dependent Claim
94 words
A process for combatting powdery mildew which comprises applying to the locus of the plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine derivative of the formula: ##SPC27## or a salt thereof, wherein R 1 and R 2 are hydrogen, lower alkyl, or lower alkenyl; R 3 is lower alkyl; R 4 is lower alkyl or lower alkenyl; X is oxygen or sulfur and R 5 is hydrogen.
Claim 4
Dependent Claim
94 words
A process for combatting powdery mildew which comprises applying to the locus of the plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine derivative of the formula: ##SPC27## or a salt thereof, wherein R 1 and R 2 are hydrogen, lower alkyl, or lower alkenyl; R 3 is lower alkyl; R 4 is lower alkyl or lower alkenyl; X is oxygen or sulfur and R 5 is hydrogen.
Claim 5
Dependent Claim
44 words
A process according to claim 2 wherein R 1 is hydrogen, allyl, ethyl, propyl or butyl; R 2 is allyl, methyl, ethyl, propyl or butyl; R 3 is methyl or ethyl; R 4 is methyl, ethyl, propyl, butyl, or amyl; and X is oxygen.
Claim 6
Dependent Claim
67 words
A process for combatting powdery mildew which comprises applying to the locus of plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine compound, or salt thereof, selected from: 2-dimethylamino-4-methyl-5-n-pentyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-n-propyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-isopropylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-amino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-n-propylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-dimethylamino-4-ethyl-5-n-butyl-6-hydroxypyrimidine; 2-diethylamino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-diethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-ethyl-6-mercaptopyrimidine; 2-dimethylamino-4-methyl-5-n-butyl-6(2-dimethylaminoethylthio)pyrimidine; and 2-dimethylamino-4-methyl-5-n-butyl-6-(2-diethylaminoethylthio)pyrimidine.
Claim 7
Dependent Claim
67 words
A process for combatting powdery mildew which comprises applying to the locus of plants or to the seeds thereof or to soil in which the seeds are to be planted, which plants are susceptible to attack by powdery mildew, a fungicidally effective amount of a systemically active pyrimidine compound, or salt thereof, selected from: 2-dimethylamino-4-methyl-5-n-pentyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-n-propyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-isopropylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-amino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-n-propylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-dimethylamino-4-ethyl-5-n-butyl-6-hydroxypyrimidine; 2-diethylamino-4-methyl-5-allyl-6-hydroxypyrimidine; 2-diethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine; 2-dimethylamino-4-methyl-5-ethyl-6-mercaptopyrimidine; 2-dimethylamino-4-methyl-5-n-butyl-6(2-dimethylaminoethylthio)pyrimidine; and 2-dimethylamino-4-methyl-5-n-butyl-6-(2-diethylaminoethylthio)pyrimidine.
Claim 8
Dependent Claim
12 words
A process according to claim 1 wherein the pyrimidine derivative is 2-dimethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine.
Claim 9
Dependent Claim
12 words
A process according to claim 1 wherein the pyrimidine derivative is 2-ethylamino-4-methyl-5-n-butyl-6-hyroxypyrimidine.
Claim 10
Dependent Claim
12 words
A process according to claim 1 wherein the plants are cucurbit plants.
Claim 11
Dependent Claim
15 words
A process according to claim 1 wherein the plants are cereal crops barley or wheat.
Claim 12
Dependent Claim
26 words
A fungicidal composition for combatting powdery mildew comprising, as a systemically active ingredient, a fungicidally effective amount of 2-ethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine and an inert carrier for said ingredient.
Claim 13
Dependent Claim
26 words
A fungicidal composition for combatting powdery mildew comprising, as a systemically active ingredient, a fungicidally effective amount of 2-ethylamino-4-methyl-5-n-butyl-6-hydroxypyrimidine and an inert carrier for said ingredient.
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USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1979-09-14 | 1980-03-15 | 1980-09-14 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1983-09-14 | 1984-03-15 | 1984-09-14 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1987-09-14 | 1988-03-15 | 1988-09-14 | $7700.00 | Window Closed / Lapsed |