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US3929791A Expired / Lapsed US ⏱️ 0.0 years remaining

2 Substituted-10{8 4-(2-oxazolidi none-lower alkyl){9 -piperazine-dibenzo{8 b,f{9 thiepins

Assignee: F Hoffmann La Roche AG
•
Filing: 1973-07-12
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Granted: 1975-12-30
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Expires: 1993-07-12
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Abstract

Abstract Dibenzothiepin derivatives of the general formula WHEREIN M, N, R1, R2, R3 and X are as hereinafter set forth, AND SALTS THEREOF AS WELL AS PROCESSES FOR THEIR MANUFACTURE ARE DISCLOSED. The end products are useful as central-depressant and neuroleptic agents.

Inventors

  • 👤 Max Gerecke
  • 👤 Jean-Pierre Kaplan
  • 👤 Emilio Kyburz

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-05 09:32
CPC Classifications
C; C07; C07D; C07D337/00; C07D337/02; C07D337/06; C07D337/10; C07D337/14; C07C; C07C323/00; C07C51/00; C07C51/347; C07C51/363

Claims Analysis

Total Claims: 12
Claim 1
Independent Claim 5 words
A COMPOUND OF THE FORMULA
Claim 2
Dependent Claim 5 words
A COMPOUND OF THE FORMULA
Claim 3
Dependent Claim 10 words
A compound in accordance with claim 1 having the formula
Claim 4
Dependent Claim 17 words
A compound in accordance with claim 2, wherein n is 2, R1 is halogen, trifluoromethyl or methyl.
Claim 5
Dependent Claim 17 words
A compound in accordance with claim 3, 3-(2-(4-(2-chloro-10, 11-dihydro-dibenzo(b,f)thiepin-10-yl)-1-piperazinyl)-ethyl)-2-oxazolidinone or a pharmaceutically acceptable acid addition salt thereof.
Claim 6
Dependent Claim 17 words
A compound in accordance with claim 3, 3-(2-(4-(10,11-dihydro-2methyl-dibenzo(b,f)thiepin-10-yl)-1-piperazinyl) -ethyl)-2-oxazolidinone or a pharmaceutically acceptable acid addition salt thereof.
Claim 7
Dependent Claim 10 words
A compound in accordance with claim 1 having the formula
Claim 8
Dependent Claim 14 words
A compound in accordance with claim 6, wherein n is 2, R1 is halogen.
Claim 9
Dependent Claim 10 words
3-(2-(4-(2-Chloro-dibenzo(b,f)thiepin-10-yl)-1-piperazinyl)-ethyl)2 -oxazolidinone or a pharmaceutically acceptable acid addition salt thereof.
Claim 10
Dependent Claim 10 words
3-(2-(4-(2-Chloro-dibenzo(b,f)thiepin-10-yl)-1-piperazinyl)-ethyl)2 -oxazolidinone or a pharmaceutically acceptable acid addition salt thereof.
Claim 11
Dependent Claim 10 words
3-(2-(4-(10,11-dihydro-2-dimethylamino-dibenzo(b,f)thiepin-10-yl)1 -piperazinyl)-ethyl)-2-oxazolidinone or a pharmaceutically acceptable acid addition salt thereof.
Claim 12
Dependent Claim 10 words
3-(2-(4-(10,11-dihydro-2-dimethylamino-dibenzo(b,f)thiepin-10-yl)1 -piperazinyl)-ethyl)-2-oxazolidinone or a pharmaceutically acceptable acid addition salt thereof.

References Cited (Backward Citations)

No citation records indexed.

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1978-12-29 1979-06-30 1979-12-30 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1982-12-29 1983-06-30 1983-12-30 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1986-12-29 1987-06-30 1987-12-30 $7700.00 Window Closed / Lapsed

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