Abstract This invention is concerened with tetrahydropyrimidinyl phenyl carbonyl acid addition salts, imidazolinyl phenyl carbonyl acid addition salts, dihydroimidazoisoindolols, tetrahydropyrimidoisoindolols, and tetrahydropyrimidoisoindolol acid addition salts which are all pharmacologically efficacious as anti-depressants. The tetrahydropyrimidinyl phenyl carbonyl acid addition salts, the tetrahydropyrimidoisoindolols and the tetrahydropyrimidoisoindolol acid addition salts are also efficacious as diuretics while the imidazolinyl phenyl carbonyl acid addition salts and the dihydroimidazoisoindolols are effficacious as anorexiants. This invention is also concerned with several processes for the preparation of these compounds.
A PROCESS FOR THE PREPARATION OF A COMPOUND HAVING THE FORMULA:
Claim 2
Dependent Claim
11 words
A PROCESS FOR THE PREPARATION OF A COMPOUND HAVING THE FORMULA:
Claim 3
Dependent Claim
25 words
A process as described in claim 1 wherein the oxidizing agent is selected from the group consisting of potassium permanganate, potassium dichromate and potassium chlorate.
Claim 4
Dependent Claim
39 words
A process as described in claim 1 wherein the oxidizing agent is selected from the group consisting of potassium permanganate, potassium dichromate and potassium chlorate; the reaction-inert solvent is water; and the reaction is conducted at about room temperature.
Claim 5
Dependent Claim
28 words
A process as described in claim 1 wherein the oxidizing agent is potassium permanganate; the reaction-inert solvent in water; and the reaction is conducted at about room temperature.