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US3843778A Expired / Lapsed US ⏱️ 0.0 years remaining

Antacids

Assignee: William H Rorer Inc
•
Filing: 1972-12-26
•
Granted: 1974-10-22
•
Expires: 1992-12-26
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Abstract

Abstract A novel process for preparing improved antacid particles is disclosed.

Inventors

  • 👤 J Buehler
  • 👤 J Diamond
  • 👤 R Joslin

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-10-24 11:55
CPC Classifications
A; A61; A61K; A61K9/00; A61K9/48; A61K9/50; A61K9/5005; A61K9/5015; A61K9/20; A61K9/2095; A61K9/0087; A61K9/0095

Claims Analysis

Total Claims: 11
Claim 1
Independent Claim 212 words
A PROCESS FOR PREPARING IMPROVED ANTACID PARTICLES WHEREIN THE WET ANTACID MATERIAL IS SELECTED FROM THE GROUP CONSISTING OF ALUMINUM HYDROXIDE, ALUMINUM HYDROXYCARBONATE, ALUMINUM MAGNESIUM GLYCINATE, CALCIUM CARBONATE, DIHYDROXY ALUMINUM AMINOACETATE MAGNESIUM ALUMINATE, MAGNESIUM CARBONATE, MAGNESIUM HYDROXIDE, MAGNESIUM OXIDE AND MAGNESIUM TRISILCATE SAID ANTACID PARTICLES HAVING A SIZE BETWEEN 0.5-300 MICRONS AND BEING COATED THEREON WITH A NON-TOXIC, INERT, SUBSTANTIALLY WATER-INSOLUBLE OIL COATING, SAID OIL BEING SELECTED FROM THE GROUP CONSISTING OF ALMOND OIL, COCONUT OIL, CORN OIL, COTTONSEED OIL, REFINED LINSEED OIL, LIGHT LIQUID PETROLATUM, HEAVY LIQUID PETROLATUM, OLEIN, OLIVE OIL, PALM OIL, PEANUT OIL, PERSIC OIL, SESAME OIL, SOYBEAN OIL AND SAFFLOWER OIL, THE PROPORTION OF OIL COATING ON SAID ANTACID PARTICLES BEING BETWEEN 1:50 AND 1:1000 BY WEIGHT OF OIL TO WET ANTACID; THE PROCESS OF WHICH COMPRISES DISPERSING AN ELECTRONEGATIVELY CHARGED POWDER SELECTED FROM THE GROUP CONSISTING OF AN ALKYL ARYL SULFONATE, AN ALKYL SULFATE, A SULFONATED AMIDE OR AMINE, A SULFATED OR SULFONATED ESTER OR ETHER, AN ALKYL SULFONATE, A DIOCTYL SULFOSUCCINATE, A HYDRATED ALUMINUM SILICATE, A SILICA PIGMENT AND A MICROFINE SILICA IN SAID OIL IN AN AMOUNT SUFFICIENT TO CHARGE THE OIL DISPERSION INTIMATELY CONTACTING THE SAID DISPERSION WITH SAID WET ANTACID AND AGITATING VIGOROUSLY TO OBTAIN A HOMOGENEOUS MIXTURE OF ALL THE MATERIALS PRESENT.
Claim 2
Dependent Claim 212 words
A PROCESS FOR PREPARING IMPROVED ANTACID PARTICLES WHEREIN THE WET ANTACID MATERIAL IS SELECTED FROM THE GROUP CONSISTING OF ALUMINUM HYDROXIDE, ALUMINUM HYDROXYCARBONATE, ALUMINUM MAGNESIUM GLYCINATE, CALCIUM CARBONATE, DIHYDROXY ALUMINUM AMINOACETATE MAGNESIUM ALUMINATE, MAGNESIUM CARBONATE, MAGNESIUM HYDROXIDE, MAGNESIUM OXIDE AND MAGNESIUM TRISILCATE SAID ANTACID PARTICLES HAVING A SIZE BETWEEN 0.5-300 MICRONS AND BEING COATED THEREON WITH A NON-TOXIC, INERT, SUBSTANTIALLY WATER-INSOLUBLE OIL COATING, SAID OIL BEING SELECTED FROM THE GROUP CONSISTING OF ALMOND OIL, COCONUT OIL, CORN OIL, COTTONSEED OIL, REFINED LINSEED OIL, LIGHT LIQUID PETROLATUM, HEAVY LIQUID PETROLATUM, OLEIN, OLIVE OIL, PALM OIL, PEANUT OIL, PERSIC OIL, SESAME OIL, SOYBEAN OIL AND SAFFLOWER OIL, THE PROPORTION OF OIL COATING ON SAID ANTACID PARTICLES BEING BETWEEN 1:50 AND 1:1000 BY WEIGHT OF OIL TO WET ANTACID; THE PROCESS OF WHICH COMPRISES DISPERSING AN ELECTRONEGATIVELY CHARGED POWDER SELECTED FROM THE GROUP CONSISTING OF AN ALKYL ARYL SULFONATE, AN ALKYL SULFATE, A SULFONATED AMIDE OR AMINE, A SULFATED OR SULFONATED ESTER OR ETHER, AN ALKYL SULFONATE, A DIOCTYL SULFOSUCCINATE, A HYDRATED ALUMINUM SILICATE, A SILICA PIGMENT AND A MICROFINE SILICA IN SAID OIL IN AN AMOUNT SUFFICIENT TO CHARGE THE OIL DISPERSION INTIMATELY CONTACTING THE SAID DISPERSION WITH SAID WET ANTACID AND AGITATING VIGOROUSLY TO OBTAIN A HOMOGENEOUS MIXTURE OF ALL THE MATERIALS PRESENT.
Claim 3
Dependent Claim 22 words
The process of claim 1 wherein the improved antacid particles are further suspended into a pharmaceutical suspension containing additional pharmaceutically accepted excipients.
Claim 4
Dependent Claim 23 words
The process of claim 1 wherein the improved antacid particles are further blended with additional pharmaceutically acceptable excipients and compressed into pharmaceutical tablets.
Claim 5
Dependent Claim 24 words
The process of claim 1 wherein the electronegatively charged powder is a silica powder and the antacid particle size is substantially between 1-50 microns.
Claim 6
Dependent Claim 48 words
The process of claim 4 where the antacid is selected from the group consisting of aluminum hydroxide, calcium carbonate and magnesium hydroxide; and the oil is selected from the group consisting of corn oil, light liquid petrolatum, heavy liquid petrolatum, olein, olive oil, peanut oil and soybean oil.
Claim 7
Dependent Claim 11 words
The process of claim 5 where the oil is corn oil.
Claim 8
Dependent Claim 12 words
The process of claim 5 where the oil is light liquid petrolatum.
Claim 9
Dependent Claim 12 words
The process of claim 5 where the oil is heavy liquid petrolatum.
Claim 10
Dependent Claim 22 words
The process of claim 7 wherein the improved antacid particles are further suspended into a pharmaceutical suspension containing additional pharmaceutically accepted excipients.
Claim 11
Dependent Claim 23 words
The process of claim 7 wherein the improved antacid particles are further blended with additional pharmaceutically acceptable excipients and compressed into pharmaceutical tablets.

References Cited (Backward Citations)

No citation records indexed.

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1977-10-21 1978-04-22 1978-10-22 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1981-10-21 1982-04-22 1982-10-22 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1985-10-21 1986-04-22 1986-10-22 $7700.00 Window Closed / Lapsed

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