US3818009A
Expired / Lapsed
US
⏱️ 0.0 years remaining
Alpha, alpha-disubstituted-5-pyrimidinemethanes
Assignee: Eli Lilly and Co
•
Filing: 1972-03-13
•
Granted: 1974-06-18
•
Expires: 1992-03-13
Abstract
Abstract There is disclosed a class of Alpha , Alpha -disubstituted-5pyrimidinemethanes and substituted methanes which are useful as fungicides, bactericides, herbicides, and plant growth regulators. Internodal elongation of plants is inhibited by treatment with a compound of this invention.
Inventors
- 👤 H Taylor
- 👤 J Davenport
- 👤 R Hackler
Bibliographic Details
Application Number
—
Jurisdiction
US
Data Source
google_patents
Last Synchronized
2026-11-03 15:02
CPC Classifications
C; C07; C07D; C07D403/00; C07D403/02; C07D403/12; C07D239/00; C07D239/02; C07D239/24; C07D239/26
Claims Analysis
Total Claims: 45
Claim 1
Independent Claim
8 words
The compound of claim 1 which is 5-diphenyl-methylpyrimidine.
Claim 2
Dependent Claim
10 words
The compound of claim 1 which is 5-( Alpha -isopropyl-4-methoxybenzyl)pyrimidine.
Claim 3
Dependent Claim
32 words
A compound of claim 1 wherein X is hydroxy, R is C2-C13 alkyl, and R'' is C2-C13 alkyl, C3-C8 cycloalkyl, or phenyl, optionally substituted with halo, trifluoromethyl, C1-C4 alkyl, or C1-C4 alkoxy.
Claim 4
Dependent Claim
11 words
The compound of claim 4 which is Alpha -isopropyl- Alpha -(4-propoxyphenyl)-5-pyrimidinemethanol.
Claim 5
Dependent Claim
11 words
The compound of claim 4 which is Alpha -(t-butyl)- Alpha -(p-tolyl)-5-pyrimidinemethanol.
Claim 6
Dependent Claim
11 words
The compound of claim 4 which is Alpha -isopropyl- Alpha -(4-methoxyphenyl)-5-pyrimidinemethanol.
Claim 7
Dependent Claim
10 words
The compound of claim 4 which is Alpha -($-ethoxy-phenyl)-Alpha -isopropyl-5-pyrimidinemethanol.
Claim 8
Dependent Claim
10 words
The compound of claim 4 which is Alpha -(4-chloro-phenyl)-Alpha -isopropyl-5-pyrimidinemethanol.
Claim 9
Dependent Claim
11 words
The compound of claim 4 which is Alpha -(t-butyl)- Alpha -(4-methoxyphenyl)-5-pyrimidinemethanol.
Claim 10
Dependent Claim
11 words
The compound of claim 4 which is Alpha -(p-cumenyl)- Alpha -isopropyl-5-pyrimidinemetahnol.
Claim 11
Dependent Claim
11 words
The compound of claim 4 which is Alpha -(3,4-dichlorophenyl)- Alpha -isopropyl15-pyrimidinemethanol.
Claim 12
Dependent Claim
10 words
The compound of claim 4 which is Alpha -(3-chloro-phenyl)-Alpha -isopropyl-5-pyrimidinemethanol.
Claim 13
Dependent Claim
11 words
The compound of claim 4 which is Alpha -cyclohexyl- Alpha -isopropyl-5-pyrimidinemethanol.
Claim 14
Dependent Claim
11 words
The compound of claim 4 which is Alpha , Alpha -bis(n-nonyl-5-pyrimidinemethanol.
Claim 15
Dependent Claim
17 words
The compound of claim 4 which is Alpha -( Alpha , Alpha , Alpha -trifluoro-m-tolyl)- Alpha -isopropyl-5-pyrimidinemethanol.
Claim 16
Dependent Claim
17 words
The compound of claim 4 which is Alpha -( Alpha , Alpha , Alpha -trifluoro-p-tolyl)- Alpha -isopropyl-5-pyrimidinemethanol.
Claim 17
Dependent Claim
29 words
A compound of claim 1 wherein X is hydroxy, R is C3-C8 cycloalkyl, and R'' is C3-C8 cycloalkyl, or phenyl, optionally substituted with C1-C4 alkyl, C1-C4 alkoxy, or halo.
Claim 18
Dependent Claim
10 words
The compound of claim 18 which is Alpha -cyclopropyl-Alpha -(p-tolyl)-5-pyrimidinemethanol.
Claim 19
Dependent Claim
10 words
The compound of claim 18 which is Alpha -(4-bromophenyl)-Alpha -cyclopropyl-5-pyrimidinemethanol.
Claim 20
Dependent Claim
11 words
The compound of claim 18 which is Alpha -cyclopropyl- Alpha -(4-fluorophenyl)-5-pyrimidinemethanol.
Claim 21
Dependent Claim
11 words
The compound of claim 18 which is Alpha -cyclobutyl- Alpha -(4-methoxyphenyl)-5-pyrimidinemethanol.
Claim 22
Dependent Claim
10 words
The compound of claim 18 which is Alpha -(4-chlorophenyl)-Alpha -cyclopropyl-5-pyrimidinemethanol.
Claim 23
Dependent Claim
11 words
The compound of claim 18 which is Alpha -cyclopropyl- Alpha -(4-methoxyphenyl-5-pyrimidinemethanol.
Claim 24
Dependent Claim
11 words
The compound of claim 18 which is Alpha -cyclohexyl- Alpha -cyclopropyl-5-pyrimidinemethanol.
Claim 25
Dependent Claim
11 words
The compound of claim 18 which is Alpha -cyclopropyl- Alpha -(p-cumenyl)-5-pyrimidinemethanol.
Claim 26
Dependent Claim
10 words
The compound of claim 18 which is Alpha -(2-chloro-phenyl)-Alpha -cyclohexyl-5-pyrimidinemethanol.
Claim 27
Dependent Claim
11 words
The compound of claim 18 which is Alpha -cyclohexyl- Alpha -(2-methoxyphenyl)-5-pyrimidinemethanol.
Claim 28
Dependent Claim
11 words
The compound of claim 18 which is Alpha -cyclohexyl- Alpha -phenyl-5-pyrimidinemethanol.
Claim 29
Dependent Claim
11 words
The compound of claim 18 which is Alpha -cyclohexyl- Alpha -(2-fluorophenyl)-5-pyrimidinemethanol.
Claim 30
Dependent Claim
11 words
The compound of claim 18 which is Alpha -cyclohexyl- Alpha -pentafluorophenyl-5-pyrimddinemethanol.
Claim 31
Dependent Claim
27 words
A compound of claim 1 wherein X is hydroxy, R is phenyl, optionally substituted with halo, and R'' is phenyl, optionally substituted with halo, or C1-C4 alkoxy.
Claim 32
Dependent Claim
10 words
The compound of claim 32 which is Alpha -(2-fluorophenyl)-Alpha -(4-fluorophenyl)-5-pyrimidinemethanol.
Claim 33
Dependent Claim
10 words
The compound of claim 32 which is Alpha -(2-chlorophenyl)-Alpha -(3-chlorophenyl-5-pyrimidinemethanol.
Claim 34
Dependent Claim
11 words
The compound of claim 32 which is Alpha , Alpha -bis(2-chlorophenyl)-5-pyrimidinemethanol.
Claim 35
Dependent Claim
11 words
The compound of claim 32 which is Alpha -(4-chlorophenyl)-Alpha -phenyl-5-pyrimidinemethanol hydrochloride.
Claim 36
Dependent Claim
10 words
The compound of claim 32 which is Alpha -(4-fluorophenyl)-Alpha -phenyl-5-pyrimidinemethanol.
Claim 37
Dependent Claim
10 words
The compound of claim 32 which is Alpha -(2-fluorophenyl)-Alpha -phenyl-5-pyrimidinemethanol.
Claim 38
Dependent Claim
10 words
The compound of claim 32 which is Alpha -(2-chlorophenyl)-Alpha -(4-fluorophenyl)-5-pyrimidinemethanol.
Claim 39
Dependent Claim
10 words
The compound of claim 32 which is Alpha -(2-fluorophenyl)-Alpha -(3-fluorophenyl)-5-pyrimidinemethanol.
Claim 40
Dependent Claim
10 words
The compound of claim 32 which is Alpha -(4-methoxyphenyl)-Alpha -phenyl-5-pyrimidinemethanol.
Claim 41
Dependent Claim
11 words
The compound of claim 32 which is Alpha -(2,5-dichlorophenyl)- Alpha -phenyl-5-pyrimidinemethanol.
Claim 42
Dependent Claim
11 words
The compound of claim 32 which is Alpha -(2,4-difluorophenyl)- Alpha -phenyl-5-pyrimidinemethanol.
Claim 43
Dependent Claim
11 words
The compound of claim 32 which is Alpha -(2,4-dichloro-phenyl)- Alpha -phenyl-5-pyrimidinemethanol.
Claim 44
Dependent Claim
10 words
The compound of claim 32 which is Alpha -(2-chlorophenyl)-Alpha -(4-methoxyphenyl)-5-pyrimidinemethanol.
Claim 45
Dependent Claim
11 words
The compound of claim 32 which is Alpha , Alpha -diphenyl-5-pyrimidinemethanol.
References Cited (Backward Citations)
US3461125A
Cited
USPTO Annuity & Maintenance Windows
| Annuity Stage | Window Opens | Payment Deadline | Surcharge Period Until | Estimated Fee | Status |
|---|---|---|---|---|---|
| 3.5 Years (Year 4) | 1977-06-17 | 1977-12-17 | 1978-06-18 | $2000.00 | Window Closed / Lapsed |
| 7.5 Years (Year 8) | 1981-06-17 | 1981-12-17 | 1982-06-18 | $3760.00 | Window Closed / Lapsed |
| 11.5 Years (Year 12) | 1985-06-17 | 1985-12-17 | 1986-06-18 | $7700.00 | Window Closed / Lapsed |