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US3719669A Expired / Lapsed US ⏱️ 0.0 years remaining

Amino(or amido)-phenyl-alkyl-benzazepine analgesics and narcotic antagonists

Assignee: Pennwalt Corp
•
Filing: 1972-03-27
•
Granted: 1973-03-06
•
Expires: 1992-03-27
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Abstract

Abstract Compounds of the general formula: D R A W I N G

Inventors

  • 👤 B Shetty

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-11-03 12:42
CPC Classifications
C; C07; C07D; C07D223/00; C07D223/14; C07D223/16

Claims Analysis

Total Claims: 21
Claim 1
Independent Claim 5 words
A compound of the formula:
Claim 2
Dependent Claim 5 words
A compound of the formula:
Claim 3
Dependent Claim 21 words
The compound of claim 1 wherein R is p-aminophenethyl; R1 is methyl and each of R2, R3 and R4 is hydrogen.
Claim 4
Dependent Claim 9 words
The compound of claim 2 which is (+)-3-(p-aminophenethyl)-2-methyl-1,2,4,5-tetrahydro-3H,3-benzazepine dihydrochloride.
Claim 5
Dependent Claim 9 words
The compound of claim 2 which is (-)-3-(p-aminophenethyl)-2-methyl-1,2,4,5-tetrahydro-3H,3-benzazepine dihydrochloride.
Claim 6
Dependent Claim 23 words
The compound of claim 1 wherein R is p-aminophenethyl; R1 is methyl; R3 is 7-hydroxy, and each of R2 and R4 is hydrogen.
Claim 7
Dependent Claim 23 words
The compound of claim 1 wherein R is p-aminophenethyl; R1 is methyl; R4 is 8-hydroxy, and each of R2 and R3 is hydrogen.
Claim 8
Dependent Claim 23 words
The compound of claim 1 wherein R is p-aminophenethyl; R1 is methyl; R3 is 7-methoxy, and each of R2 and R4 is hydrogen.
Claim 9
Dependent Claim 23 words
The compound of claim 1 wherein R is p-aminophenethyl; R1 is methyl; R4 is 8-methoxy, and each of R2 and R3 is hydrogen.
Claim 10
Dependent Claim 9 words
The compound of claim 8 which is (-)-3-(p-aminophenethyl)-8-methoxy-2-methyl-1,2,4,5-tetrahydro-3H,3 -benzazepine.
Claim 11
Dependent Claim 9 words
The compound of claim 8 which is (+)-3-(p-aminophenethyl)-8-methoxy-2-methyl-1,2,4,5-tetrahydro-3H,3 -benzazepine.
Claim 12
Dependent Claim 21 words
The compound of claim 1 wherein R is p-aminophenethyl; each of R1, R2 and R4 is hydrogen, and R3 is 7-methoxy.
Claim 13
Dependent Claim 10 words
The compound of claim 11 which is 3-(para-amino phenyl-ethyl)-7-methoxy-1,2,4,5-tetrahydro-3H,3-benzazepine dihydrochloride.
Claim 14
Dependent Claim 21 words
The compound of claim 1 wherein R is p-aminophenethyl; each of R1, R2 and R4 is hydrogen, and R3 is 7-hydroxy.
Claim 15
Dependent Claim 10 words
The compound of claim 1 which is 3-(2-p-aminophenyl-1-methyl-ethyl)-7-methoxy-1,2,4,5-tetrahydro-3H,3 -benzazepine dihydrochloride.
Claim 16
Dependent Claim 19 words
The compound of claim 1 wherein R is p-aminophenethyl and each of R1, R2, R3 and R4 is hydrogen.
Claim 17
Dependent Claim 8 words
The compound of claim 1 which is 3-(p-acetamidophenethyl)-1-,2,4,5-tetrahydro-3H,3-benzazepine.
Claim 18
Dependent Claim 21 words
The compound of claim 1 wherein R is p-acetamidophenethyl; each of R1, R2 and R4 is hydrogen, and R3 is 7-hydroxy.
Claim 19
Dependent Claim 21 words
The compound of claim 1 wherein R is p-acetamidophenethyl; each of R1, R2 and R4 is hydrogen, and R3 is 7-methoxy.
Claim 20
Dependent Claim 9 words
The compound of claim 18 which is 7-methoxy-3-(p-acetamidophenethyl)-1,2,4,5-tetrahydro-3H,3-benzazepine hydrochloride.
Claim 21
Dependent Claim 23 words
The compound of claim 1 wherein R is p-acetamidophenethyl; R1 is methyl; each of R2 and R3 is hydrogen, and R4 is 8-methoxy.

References Cited (Backward Citations)

No citation records indexed.

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1976-03-05 1976-09-04 1977-03-06 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1980-03-05 1980-09-04 1981-03-06 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1984-03-05 1984-09-04 1985-03-06 $7700.00 Window Closed / Lapsed

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