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US3119742A Expired / Lapsed US ⏱️ 0.0 years remaining

Method of preparing sustained release pharmaceutical pellets and product thereof

Assignee: Smith Kline & French Laboratories Ltd
•
Filing: 1962-12-19
•
Granted: 1964-01-28
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Expires: 1982-12-19
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Abstract

No abstract record available.

Inventors

  • 👤 Kenneth R Heimlich
  • 👤 Donald R Macdonnell

Bibliographic Details

Application Number —
Jurisdiction US
Data Source google_patents
Last Synchronized 2026-10-23 12:41
CPC Classifications
A; A61; A61J; A61J3/00; A61J3/005; A61K; A61K9/00; A61K9/48; A61K9/50; A61K9/5005; A61K9/5015; A61K9/5084

Claims Analysis

Total Claims: 2
Claim 1
Independent Claim 109 words
THE METHOD OF PREPARING SUSTAINED RELEASE ORALLY ADMINISTRABLE PHARMACEUTICAL PELLETS CONTAINING A UNIT DOSAGE AMOUNT OF FROM ABOUT 200 MG. TO ABOUT 600 MG. OF A HIGH DOSAGE MEDICAMENT WHICH COMPRISES; (A) WETTING A MEDICAMENT IN SUBSTANTIALLY SPHERICAL CRYSTALLINE FORM ROTATING IN A COATING PAN WITH AN ADHESIVE SOLUTION. (B) COATING SAID WETTED CRYSTALLINE MEDICAMENT WITH ADDITIONAL POWDERED MEDICAMENT TO FORM SUBSTANTIALLY SMOOTH, SPHERICAL PELLETS. (C) DRYING AND SEPARATING SAID PELLETS INTO A PLURALITY OF GROUPS, (D) COATING AT LEAST ONE OF SAID GROUPS OF PELLETS WITH A PHARMACEUTICALLY ACCEPTABLE SUSTAINED RELEASE LIPID MATERIAL RESISTANT TO DISINTEGRATION AND SLOWLY DISPERSIBLE IN THE GASTROINTESTINAL TRACT, AND (E) BLENDING SAID GROUPS.
Claim 2
Independent Claim 109 words
THE METHOD OF PREPARING SUSTAINED RELEASE ORALLY ADMINISTRABLE PHARMACEUTICAL PELLETS CONTAINING A UNIT DOSAGE AMOUNT OF FROM ABOUT 200 MG. TO ABOUT 600 MG. OF A HIGH DOSAGE MEDICAMENT WHICH COMPRISES; (A) WETTING A MEDICAMENT IN SUBSTANTIALLY SPHERICAL CRYSTALLINE FORM ROTATING IN A COATING PAN WITH AN ADHESIVE SOLUTION. (B) COATING SAID WETTED CRYSTALLINE MEDICAMENT WITH ADDITIONAL POWDERED MEDICAMENT TO FORM SUBSTANTIALLY SMOOTH, SPHERICAL PELLETS. (C) DRYING AND SEPARATING SAID PELLETS INTO A PLURALITY OF GROUPS, (D) COATING AT LEAST ONE OF SAID GROUPS OF PELLETS WITH A PHARMACEUTICALLY ACCEPTABLE SUSTAINED RELEASE LIPID MATERIAL RESISTANT TO DISINTEGRATION AND SLOWLY DISPERSIBLE IN THE GASTROINTESTINAL TRACT, AND (E) BLENDING SAID GROUPS.

References Cited (Backward Citations)

US2738303A Cited
US2793979A Cited
US2921883A Cited

USPTO Annuity & Maintenance Windows

Annuity Stage Window Opens Payment Deadline Surcharge Period Until Estimated Fee Status
3.5 Years (Year 4) 1967-01-27 1967-07-29 1968-01-28 $2000.00 Window Closed / Lapsed
7.5 Years (Year 8) 1971-01-27 1971-07-29 1972-01-28 $3760.00 Window Closed / Lapsed
11.5 Years (Year 12) 1975-01-27 1975-07-29 1976-01-28 $7700.00 Window Closed / Lapsed

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