GB2042535A
Expired / Lapsed
GB
⏱️ 0.0 years remaining
1-acylated-1,2,3,4-tetrahydroquinoline-2-carboxylic acids
Assignee: ATK Launch Systems LLC
•
Filing: 1980-02-05
•
Granted: —
•
Expires: 2000-02-05
Abstract
No abstract record available.
Inventors
No inventors recorded.
Bibliographic Details
Application Number
—
Jurisdiction
GB
Data Source
google_patents
Last Synchronized
2026-10-23 04:10
CPC Classifications
C; C07; C07D; C07D215/00; C07D215/02; C07D215/16; C07D215/48
Claims Analysis
Total Claims: 80
Claim 1
Independent Claim
70 words
A compound of the formula: R R3 2-, R 14 Rl-S-(H2)M-L M - -N 0 COOH wherein R, is benzoyl, acetyl, hydrogen or R R3 2-, R 14 -S-CHI-CH-C-N 11 0n CODH (1) GB 2 042 535 A R2 is hydrogen, methoxy or methyl; R3 is hydrogen, methoxy, methyl, chloro or hydroxy; R4 is hydrogen, methyl or acetyithiomethyi; m is 0 or 1, and the sodium and dicyclohexylamine salts thereof.
Claim 2
Dependent Claim
70 words
A compound of the formula: R R3 2-, R 14 Rl-S-(H2)M-L M - -N 0 COOH wherein R, is benzoyl, acetyl, hydrogen or R R3 2-, R 14 -S-CHI-CH-C-N 11 0n CODH (1) GB 2 042 535 A R2 is hydrogen, methoxy or methyl; R3 is hydrogen, methoxy, methyl, chloro or hydroxy; R4 is hydrogen, methyl or acetyithiomethyi; m is 0 or 1, and the sodium and dicyclohexylamine salts thereof.
Claim 3
Dependent Claim
6 words
The dicyclohexylamine salt of 1-[(3-benzoyithio)-1-oxopropyll-1,2,3,4tetrahydroquinoline-2carboxylic acid.
Claim 4
Dependent Claim
6 words
The dicyclohexylamine salt of 1-[(3-benzoyithio)-1-oxopropyll-1,2,3,4tetrahydroquinoline-2carboxylic acid.
Claim 5
Dependent Claim
7 words
The sodium salt of 1-[(3-benzoylthio)-1-oxopropyll-1,2,3,4tetrahydroquinoline-2-carboxyiic acid. 5
Claim 6
Dependent Claim
7 words
The sodium salt of 1-[(3-benzoylthio)-1-oxopropyll-1,2,3,4tetrahydroquinoline-2-carboxyiic acid. 5
Claim 7
Dependent Claim
7 words
The dicyclohexylamine salt of 1,2,3,4-tetrahydro-l-[(3-mercapto)-1- oxopropyll-quinoline-2-carboxylic acid.
Claim 8
Dependent Claim
7 words
The dicyclohexylamine salt of 1,2,3,4-tetrahydro-l-[(3-mercapto)-1- oxopropyll-quinoline-2-carboxylic acid.
Claim 9
Dependent Claim
3 words
( )-1-(3-Benzoyithio-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 10
Dependent Claim
3 words
( )-1-(3-Benzoyithio-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 11
Dependent Claim
9 words
The dicyclohexylamine salt of (S) (-)-1-(3)benzoyithio-l-oxopropyi)-1,2, 3,4-tetrahydro-2- quinolinecarboxylic acid.
Claim 12
Dependent Claim
9 words
The dicyclohexylamine salt of (S) (-)-1-(3)benzoyithio-l-oxopropyi)-1,2, 3,4-tetrahydro-2- quinolinecarboxylic acid.
Claim 13
Dependent Claim
3 words
(S)(-)-1-(3-Benzoyithio-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarboxyli c acid.
Claim 14
Dependent Claim
3 words
(S)(-)-1-(3-Benzoyithio-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarboxyli c acid.
Claim 15
Dependent Claim
7 words
The sodium salt of (S)(-)-1-(3-benzoyithiol-oxopropyi)-1,2,3,4tetrahydro-2-quinolinecarboxyli c acid.
Claim 16
Dependent Claim
7 words
The sodium salt of (S)(-)-1-(3-benzoyithiol-oxopropyi)-1,2,3,4tetrahydro-2-quinolinecarboxyli c acid.
Claim 17
Dependent Claim
10 words
The dicycl ohexyla mine salt of (R)(+)-1 - (3-benzoylthio-l-oxopropyl)1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 18
Dependent Claim
10 words
The dicycl ohexyla mine salt of (R)(+)-1 - (3-benzoylthio-l-oxopropyl)1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 19
Dependent Claim
17 words
The sodium salt of (R) W-11 -(3-benzoylth io- 1 -oxo pro pyi)-1,2,3,4tetrahydro-2-q ui no] inecarboxyl ic acid.
Claim 20
Dependent Claim
17 words
The sodium salt of (R) W-11 -(3-benzoylth io- 1 -oxo pro pyi)-1,2,3,4tetrahydro-2-q ui no] inecarboxyl ic acid.
Claim 21
Dependent Claim
3 words
( )-1-(3-Acetyithio-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 22
Dependent Claim
3 words
( )-1-(3-Acetyithio-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 23
Dependent Claim
19 words
The sodium salt of (S) (-)-1 -(3-acetylthio-1 -oxo pro pyl)-1,2,3,4tetrahyd ro-2-q u ino 1 i neca rboxyl ic acid.
Claim 24
Dependent Claim
19 words
The sodium salt of (S) (-)-1 -(3-acetylthio-1 -oxo pro pyl)-1,2,3,4tetrahyd ro-2-q u ino 1 i neca rboxyl ic acid.
Claim 25
Dependent Claim
2 words
(S)(-)-1-(3-Acetyithio-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 26
Dependent Claim
2 words
(S)(-)-1-(3-Acetyithio-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 27
Dependent Claim
15 words
( )-1-(3-Merca pto-1 -oxo pro pyi)-1,2,3,4-tetra hyd ro-2-qu i nol i neca rboxyl ic acid.
Claim 28
Dependent Claim
15 words
( )-1-(3-Merca pto-1 -oxo pro pyi)-1,2,3,4-tetra hyd ro-2-qu i nol i neca rboxyl ic acid.
Claim 29
Dependent Claim
9 words
The sodium salt of ( )-1 -(3-mereapto-1 -oxopropyi)-1,2,3,4tetrahydro-2-quinolinecarboxylic acid.
Claim 30
Dependent Claim
9 words
The sodium salt of ( )-1 -(3-mereapto-1 -oxopropyi)-1,2,3,4tetrahydro-2-quinolinecarboxylic acid.
Claim 31
Dependent Claim
18 words
(S) (+1 -(3-M erca pto-1 -oxo pro pyl)-1,2,3,4-tetra hyd ro-2-q u i no 1 ineca rboxyl ic acid.
Claim 32
Dependent Claim
18 words
(S) (+1 -(3-M erca pto-1 -oxo pro pyl)-1,2,3,4-tetra hyd ro-2-q u i no 1 ineca rboxyl ic acid.
Claim 33
Dependent Claim
17 words
( ) 1,1'-[Dithiobis(l -oxo-3,1 -pro pa nediyi 1-bis- 1,2,3,4-tetra hydro-2-q u i no 1 i necarboxylic acid.
Claim 34
Dependent Claim
17 words
( ) 1,1'-[Dithiobis(l -oxo-3,1 -pro pa nediyi 1-bis- 1,2,3,4-tetra hydro-2-q u i no 1 i necarboxylic acid.
Claim 35
Dependent Claim
16 words
( )-1 -(3-Benzoylth lo-2-m ethy]-1 -oxo pro pyl)-1,2,3,4-tetrahyd ro2-q u in ol i necarboxyl ic acid.
Claim 36
Dependent Claim
16 words
( )-1 -(3-Benzoylth lo-2-m ethy]-1 -oxo pro pyl)-1,2,3,4-tetrahyd ro2-q u in ol i necarboxyl ic acid.
Claim 37
Dependent Claim
13 words
The dicyclohexylamine salt of ( )-1 -(3-acetylthio-2-methyi-l -oxo pro pyl)-1,2,3,4-tetrahyd ro-2- quinolinecarboxylic acid.
Claim 38
Dependent Claim
13 words
The dicyclohexylamine salt of ( )-1 -(3-acetylthio-2-methyi-l -oxo pro pyl)-1,2,3,4-tetrahyd ro-2- quinolinecarboxylic acid.
Claim 39
Dependent Claim
4 words
( )-1-(3)Acetyithio-2-methyi-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarbo xylic acid.
Claim 40
Dependent Claim
4 words
( )-1-(3)Acetyithio-2-methyi-l-oxopropyi)-1,2,3,4-tetrahydro-2quinolinecarbo xylic acid.
Claim 41
Dependent Claim
14 words
( )-1-(3-Acetylth io-2-acetylth lomethyl- 1 -oxo pro pyi)-1,2,3,4tetrahydro-2-q ui nol i necarboxyl ic acid.
Claim 42
Dependent Claim
14 words
( )-1-(3-Acetylth io-2-acetylth lomethyl- 1 -oxo pro pyi)-1,2,3,4tetrahydro-2-q ui nol i necarboxyl ic acid.
Claim 43
Dependent Claim
16 words
(-)-1-[(2R)-3-Acetylth io-2-m ethyl -1 -oxo pro pyl 1-(2S)- 1,2,3,4tetra hydro-2-qu i noi i necarboxyl ic acid.
Claim 44
Dependent Claim
16 words
(-)-1-[(2R)-3-Acetylth io-2-m ethyl -1 -oxo pro pyl 1-(2S)- 1,2,3,4tetra hydro-2-qu i noi i necarboxyl ic acid.
Claim 45
Dependent Claim
4 words
(-)-1-[(2S)-Acetyithio-2-methyi-l-oxopropyll-(2S)-1,2,3,4-tetrahydro2-quino linecarboxylic acid. 30
Claim 46
Dependent Claim
4 words
(-)-1-[(2S)-Acetyithio-2-methyi-l-oxopropyll-(2S)-1,2,3,4-tetrahydro2-quino linecarboxylic acid. 30
Claim 47
Dependent Claim
4 words
( )-1-(3-Mercapto-2-methyi-l-oxopropyl)-1,2,3,4-tetrahydro-2quinolinecarboxy iic acid.
Claim 48
Dependent Claim
4 words
( )-1-(3-Mercapto-2-methyi-l-oxopropyl)-1,2,3,4-tetrahydro-2quinolinecarboxy iic acid.
Claim 49
Dependent Claim
3 words
( )-1-(2-Benzoyithio-l-oxoethyl-1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 50
Dependent Claim
3 words
( )-1-(2-Benzoyithio-l-oxoethyl-1,2,3,4-tetrahydro-2quinolinecarboxylic acid.
Claim 51
Dependent Claim
8 words
The dicyclohexyiamine salt of ( )-1-(2-Mercapto-l-oxoethyi)-1,2,3,4tetrahydro2- quinolinecarboxylic acid.
Claim 52
Dependent Claim
8 words
The dicyclohexyiamine salt of ( )-1-(2-Mercapto-l-oxoethyi)-1,2,3,4tetrahydro2- quinolinecarboxylic acid.
Claim 53
Dependent Claim
8 words
The sodium salt of ( )-1-(2-mercapto-l-oxoethyi)-1,2,3,4-tetrahydro-2quinolinecarboxylic acid. 35
Claim 54
Dependent Claim
8 words
The sodium salt of ( )-1-(2-mercapto-l-oxoethyi)-1,2,3,4-tetrahydro-2quinolinecarboxylic acid. 35
Claim 55
Dependent Claim
4 words
( )-1-(2-Mercapto-l-oxoethyi)-1,2,3,4-tetrahydro-2- quinolinecarboxylic acid.
Claim 56
Dependent Claim
4 words
( )-1-(2-Mercapto-l-oxoethyi)-1,2,3,4-tetrahydro-2- quinolinecarboxylic acid.
Claim 57
Dependent Claim
4 words
( )-1,1'[Dithiobis(l-oxo-2,1-ethanediyi)l-bis-1,2,3,4-tetrahydro-2qulnolinec arboxylic acid.
Claim 58
Dependent Claim
4 words
( )-1,1'[Dithiobis(l-oxo-2,1-ethanediyi)l-bis-1,2,3,4-tetrahydro-2qulnolinec arboxylic acid.
Claim 59
Dependent Claim
16 words
( )-1 -(2-Benzoyith io-1 -oxo pro pyi)-1,2,3,4-tetrahyd ro-2-q u in o 1 i necarboxyl ic acid.
Claim 60
Dependent Claim
16 words
( )-1 -(2-Benzoyith io-1 -oxo pro pyi)-1,2,3,4-tetrahyd ro-2-q u in o 1 i necarboxyl ic acid.
Claim 61
Dependent Claim
19 words
( )-1 -(2-Me rca pto- 1 -oxo pro pyi)- 1,2,3,4-tetrahyd ro-2-q u in o 1 i necarboxyl ic acid.
Claim 62
Dependent Claim
19 words
( )-1 -(2-Me rca pto- 1 -oxo pro pyi)- 1,2,3,4-tetrahyd ro-2-q u in o 1 i necarboxyl ic acid.
Claim 63
Dependent Claim
4 words
( )-1-(3-Benzoyithio-l-oxopropyi-1,2,3,4-tetrahydro-6-methoxy-2quinolinecarb oxylic acid.
Claim 64
Dependent Claim
4 words
( )-1-(3-Benzoyithio-l-oxopropyi-1,2,3,4-tetrahydro-6-methoxy-2quinolinecarb oxylic acid.
Claim 65
Dependent Claim
8 words
The dicyclohexylamine salt of ( )-1-(3-mercapto-l-oxopropyi)-1,2,3,4tetrahydro-6-methoxy-2- quinolinecarboxylic acid.
Claim 66
Dependent Claim
8 words
The dicyclohexylamine salt of ( )-1-(3-mercapto-l-oxopropyi)-1,2,3,4tetrahydro-6-methoxy-2- quinolinecarboxylic acid.
Claim 67
Dependent Claim
4 words
( )-1-(3-Acetyithio-l-oxopropyi)-1,2,3,4-tetrahydro-6,7-dimethoxy-2quinoline carboxylic acid.
Claim 68
Dependent Claim
4 words
( )-1-(3-Acetyithio-l-oxopropyi)-1,2,3,4-tetrahydro-6,7-dimethoxy-2quinoline carboxylic acid.
Claim 69
Dependent Claim
4 words
( )-1-(2-Acetylthio-l-oxopropyi)-1,2,3,4-tetrahydro-6-methyl-2quinolinecarbo xylic acid.
Claim 70
Dependent Claim
4 words
( )-1-(2-Acetylthio-l-oxopropyi)-1,2,3,4-tetrahydro-6-methyl-2quinolinecarbo xylic acid.
Claim 71
Dependent Claim
10 words
The dicyclohexylamine salt of ( )-1-(3-acetyithio-l-oxopropyi)-1,2,3, 4-tetrahydro-7-methyi-2- 45 quinolinecarboxylic acid.
Claim 72
Dependent Claim
10 words
The dicyclohexylamine salt of ( )-1-(3-acetyithio-l-oxopropyi)-1,2,3, 4-tetrahydro-7-methyi-2- 45 quinolinecarboxylic acid.
Claim 73
Dependent Claim
4 words
( )-1-(3-Acetylthio-l-oxopropyi)-1,2,3,4-tetrahydro-7-methyi-2quinolinecarbo xylic acid.
Claim 74
Dependent Claim
4 words
( )-1-(3-Acetylthio-l-oxopropyi)-1,2,3,4-tetrahydro-7-methyi-2quinolinecarbo xylic acid.
Claim 75
Dependent Claim
4 words
( )-1-(3-Acetyithio-l-oxopropyl)-6-chloro-1,2,3,4-tetrahydro-2quinolinecarbo xylic acid.
Claim 76
Dependent Claim
4 words
( )-1-(3-Acetyithio-l-oxopropyl)-6-chloro-1,2,3,4-tetrahydro-2quinolinecarbo xylic acid.
Claim 77
Dependent Claim
13 words
( )-1-(3-Acetyithio-l-oxo pro pyi)- 1,2,3,4-tetra hydro-6-hyd roxy-2qu inol i neca rboxyl ic acid.
Claim 78
Dependent Claim
13 words
( )-1-(3-Acetyithio-l-oxo pro pyi)- 1,2,3,4-tetra hydro-6-hyd roxy-2qu inol i neca rboxyl ic acid.
Claim 79
Dependent Claim
28 words
A pharmaceutical composition for human or veterinary use comprising at least one compound 50 according to any of claims 1 to 39 and an inert, pharmaceutically acceptable carrier.
Claim 80
Dependent Claim
52 words
A composition according to claim 40 in dosage unit form, each dosage unit containing 10 to 500 mg of said compound(s). Printed for Her Majesty's Stationery Office, by Croydon Printing Company Limited, Croydon Surrey, 1980. Published by the Patent Office, 25 Southampton Buildings, London, WC2A lAY, from which copies may be obtained.
References Cited (Backward Citations)
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